| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5271498 | 13 | ID50 | = | 58 | uM | ALA5230918 | uM | Homo sapiens | |||
| 2. |  ALA5274402 | 11 | ID50 | = | 18 | uM | ALA5230918 | uM | Homo sapiens | |||
| 3. |  ALA4169569 | 10 | Activity | = | 38.8 | % | ALA4155369 | % | Homo sapiens | |||
| 4. |  TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 5. |  GSK1059615 | GSK-1059615 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 6. |  ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 7. |  CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 8. |  JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 9. |  Saracatinib (AZD0530) | 33, AZD-0530 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 10. |  Tandutinib (MLN518) | 75 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 11. |  Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 12. |  Cabozantinib (XL184, BMS-907351) | CABOZANTINIB | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 13. |  RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 14. |  Ravoxertinib | RAVOXERTINIB | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 15. |  Flavopiridol | 1 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 16. |  BAY 80-6946 (Copanlisib) | 46, BAY80-6946 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 17. |  Pexidartinib | PEXIDARTINIB | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 18. |  GSK461364 | GSK-461364A | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 19. |  PF-04691502 | 3 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens | ||
| 20. |  MLN2480 | SID174006384 | Kd apparent | > | 30000 | nM | ALA3991687 | Inactive | nM | Homo sapiens |
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