# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Adenosine 3',5'-Cyclic Monophosphate Sodium Salt Hydrate | SID56320726 | EC50 | = | 5.62 | uM | ALA4402333 | 5.25 | nM | Homo sapiens | ||
2. | 8-Bromo-cAMP sodium salt | NCGC00093662-01 | EC50 | = | 1.09 | uM | ALA4402333 | 5.96 | nM | Homo sapiens | ||
3. | ALA4468490 | 7C-cAMP | EC50 | = | 2.75 | uM | ALA4402333 | 5.56 | nM | Homo sapiens | ||
4. | ALA4549036 | 8Br-7C-cAMP | EC50 | = | 0.53 | uM | ALA4402333 | 6.28 | nM | Homo sapiens | ||
5. | ALA4442766 | 7Br-7C-cAMP | EC50 | = | 2.54 | uM | ALA4402333 | 5.59 | nM | Homo sapiens | ||
6. | ESI 09 | 23, ESI-09 | Activity | <= | 20 | % | ALA4397756 | % | Homo sapiens | |||
7. | ESI 09 | 23, ESI-09 | Activity | = | 44 | % | ALA4397755 | % | Homo sapiens | |||
8. | ESI 09 | 23, ESI-09 | Activity | = | 30 | % | ALA4397754 | % | Homo sapiens | |||
9. | ESI 09 | 23, ESI-09 | Activity | 0 | ALA4397753 | Not Active | Homo sapiens | |||||
10. | (R)-CE3F4 | 12a; R-CE3F4 | Ratio | = | 5 | ALA4397753 | Homo sapiens | |||||
11. | (R)-CE3F4 | 12a; R-CE3F4 | Kd(app) | = | 757 | uM | ALA4397752 | nM | Homo sapiens | |||
12. | (R)-CE3F4 | 12a; R-CE3F4 | Kd | = | 124 | uM | ALA4397751 | nM | Homo sapiens | |||
13. | ESI 09 | 23, ESI-09 | Activity | 0 | ALA4397735 | Active | Homo sapiens | |||||
14. | ESI 09 | 23, ESI-09 | Activity | 0 | ALA4397731 | Active | Homo sapiens | |||||
15. | ESI 09 | 23, ESI-09 | Activity | 0 | ALA4397698 | Active | Homo sapiens | |||||
16. | (R)-CE3F4 | 12a; R-CE3F4 | Activity | 0 | ALA4397699 | Not Active | Homo sapiens | |||||
17. | (R)-CE3F4 | 12a; R-CE3F4 | Activity | 0 | ALA4397729 | Active | Homo sapiens | |||||
18. | ESI 09 | 23, ESI-09 | Activity | = | 250 | nm | ALA4397727 | nm | Homo sapiens | |||
19. | ESI 09 | 23, ESI-09 | Activity | <= | 5 | nm | ALA4397726 | nm | Homo sapiens | |||
20. | ESI 09 | 23, ESI-09 | Kd | = | 20 | uM | ALA4397718 | 4.70 | nM | Homo sapiens |