| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  5-Hydroxyindole | 16 | Kd | = | 2.1 | mM | ALA3430212 | 2.68 | nM | Homo sapiens | ||
| 2. |  (S)-2-Amino-3-(1H-indol-3-yl)-propionic acid methyl ester | 77 | Kd | = | 570 | uM | ALA3430212 | 3.24 | nM | Homo sapiens | ||
| 3. |  ALA3427779 | 20 | Kd | = | 35 | uM | ALA3430212 | 4.46 | nM | Homo sapiens | ||
| 4. |  ALA3427780 | 21 | Kd | = | 3 | uM | ALA3430212 | 5.52 | nM | Homo sapiens | ||
| 5. |  ALA3427781 | 22 | Kd | = | 1.3 | uM | ALA3430212 | 5.89 | nM | Homo sapiens | ||
| 6. |  ALA3415473 | IBR120 (R) | INH | 0 | ALA3420715 | Active | % | Homo sapiens | ||||
| 7. |  IBR2 | 6, IBR2 | INH | 0 | ALA3420716 | Active | % | Homo sapiens | ||||
| 8. | ALA3415473 | IBR120 (R) | INH | 0 | ALA3420717 | Dose-dependent effect | % | Homo sapiens | ||||
| 9. | IBR2 | 6, IBR2 | INH | 0 | ALA3420718 | Active | % | Homo sapiens | ||||
| 10. |  B02 | SID24787209 | FC | = | 4 | ALA3377964 | Homo sapiens | |||||
| 11. | B02 | SID24787209 | FC | = | 8 | ALA3377963 | Homo sapiens | |||||
| 12. | IBR2 | 6, IBR2 | FC | = | 2 | ALA3377962 | Homo sapiens | |||||
| 13. | IBR2 | 6, IBR2 | FC | = | 10 | ALA3377961 | Homo sapiens | |||||
| 14. |  4-Bromo-N-(4-bromophenyl)-3-[[(phenylmethyl)amino]sulfonyl]benzamide | SID24416418 | FC | = | 1.5 | ALA3377960 | Homo sapiens | |||||
| 15. |  ALA4559055 | 27 | Activity | = | 24 | % | ALA4480879 | % | Homo sapiens | |||
| 16. |  ALA4530772 | 26 | Activity | = | 40 | % | ALA4480878 | % | Homo sapiens | |||
| 17. |  ALA4577556 | 2 | Activity | 0 | ALA4480877 | Not Active | Homo sapiens | |||||
| 18. |  ALA4549046 | 42 | EC50 | 0 | ALA4480875 | Not Active | Homo sapiens | |||||
| 19. |  ALA4576696 | 1 | EC50 | = | 53 | uM | ALA4480875 | 4.28 | nM | Homo sapiens | ||
| 20. | ALA4577556 | 2 | EC50 | = | 25 | uM | ALA4480875 | 4.60 | nM | Homo sapiens |
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