| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  dilazep | Dilazep | IC50 | > | 50 | uM | ALA2077530 | inhibitor [IC50>50uM] | nM | Homo sapiens | ||
| 2. |  Sildenafil | 1 | IC50 | = | 80 | uM | ALA2077530 | 4.10 | inhibitor [IC50=80uM] | nM | Homo sapiens | |
| 3. |  MK 571 sodium salt (L 660711 sodium salt) | Mk-679 | IC50 | = | 40 | uM | ALA2077530 | 4.40 | inhibitor [IC50=40uM] | nM | Homo sapiens | |
| 4. |  Dipyridamole | Dipyridamole | IC50 | = | 30 | uM | ALA2077530 | 4.52 | inhibitor [IC50=30uM] | nM | Homo sapiens | |
| 5. |  ALA285913 | Trequinsin | IC50 | = | 30 | uM | ALA2077530 | 4.52 | inhibitor [IC50=30uM] | nM | Homo sapiens | |
| 6. |  ALA832 | Sulfinpyrazone | IC50 | < | 100 | uM | ALA2078531 | inhibitor [IC50=<100 uM] | nM | Homo sapiens | ||
| 7. |  Adenosine 3′,5′-cyclic monophosphate | Cyclic AMP | Km | = | 379 | uM | ALA2075979 | substrate [Km=379uM] | nM | Homo sapiens | ||
| 8. |  Guanosine 3′,5′-cyclic monophosphate | cGMP | Km | = | 2.1 | uM | ALA2075979 | substrate [Km=2.1uM] | nM | Homo sapiens | ||
| 9. |  Thromboxane B2 | SID26754848 | Activity | = | 77 | % | ALA2078526 | inhibitor [77% of control] | % | Homo sapiens | ||
| 10. |  Prostaglandin E₂ | PGE2 | Activity | = | 74 | % | ALA2078528 | inhibitor [74% of control] | % | Homo sapiens | ||
| 11. |  Prostaglandin E1 | PGE1 | Activity | = | 69 | % | ALA2078529 | inhibitor [69% of control] | % | Homo sapiens | ||
| 12. |  Dinoprost | 9 | Activity | = | 63 | % | ALA2078527 | inhibitor [63% of control] | % | Homo sapiens | ||
| 13. | Guanosine 3′,5′-cyclic monophosphate | cGMP | Activity | = | 37 | % | ALA2075980 | inhibitor [37 % of control] | % | Homo sapiens | ||
| 14. | Adenosine 3′,5′-cyclic monophosphate | Cyclic AMP | Activity | = | 35.5 | % | ALA2078520 | inhibitor [35.5 % of control] | % | Homo sapiens | ||
| 15. | ALA285913 | Trequinsin | Activity | = | 26.2 | % | ALA2078522 | inhibitor [26.2 % of control] | % | Homo sapiens | ||
| 16. | Sildenafil | 1 | Activity | = | 22 | % | ALA2078523 | inhibitor [22 % of control] | % | Homo sapiens | ||
| 17. |  ALA28079 | M&B-22948 | Activity | = | 12 | % | ALA2075980 | inhibitor [12 % of control] | % | Homo sapiens | ||
| 18. |  Fluorescein diacetate | SID17514836 | Activity | = | 49.2 | % | ALA2078525 | inhibitor [49.2 % of control] | % | Homo sapiens | ||
| 19. |  Prostaglandin A1 | 44, PGA1 | Activity | = | 51 | % | ALA2078530 | inhibitor [51% of control] | % | Homo sapiens | ||
| 20. | ALA28079 | M&B-22948 | Activity | = | 41 | % | ALA2078521 | inhibitor [41 % of control] | % | Homo sapiens |
The page will load shortly, Thanks for your patience!