# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4749391 | 17 | IC50 | = | 7.8 | nM | ALA4704018 | 8.11 | nM | Mus musculus | ||
2. | ALA4755139 | 16 | IC50 | = | 7.7 | nM | ALA4704018 | 8.11 | nM | Mus musculus | ||
3. | ALA4764430 | 15 | IC50 | = | 5.5 | nM | ALA4704018 | 8.26 | nM | Mus musculus | ||
4. | ALA4789376 | 14 | IC50 | = | 6.7 | nM | ALA4704018 | 8.17 | nM | Mus musculus | ||
5. | ALA4756869 | 13 | IC50 | = | 1 | nM | ALA4704018 | 9.00 | nM | Mus musculus | ||
6. | ALA4794014 | 12 | IC50 | = | 2.1 | nM | ALA4704018 | 8.68 | nM | Mus musculus | ||
7. | ALA4776610 | 11 | IC50 | = | 1.3 | nM | ALA4704018 | 8.89 | nM | Mus musculus | ||
8. | ALA4742167 | 10 | IC50 | = | 1000 | nM | ALA4704018 | 6.00 | nM | Mus musculus | ||
9. | GLPG4716 | 9; OATD-01 | Ki | = | 5.7 | nM | ALA4704018 | 8.24 | nM | Mus musculus | ||
10. | GLPG4716 | 9; OATD-01 | IC50 | = | 7.8 | nM | ALA4704018 | 8.11 | nM | Mus musculus | ||
11. | ALA4758240 | 8 | IC50 | = | 660 | nM | ALA4704018 | 6.18 | nM | Mus musculus | ||
12. | ALA4758850 | 7 | IC50 | = | 22000 | nM | ALA4704018 | 4.66 | nM | Mus musculus | ||
13. | ALA4209364 | 1 | IC50 | = | 7600 | nM | ALA4704018 | 5.12 | nM | Mus musculus | ||
14. | ALA4791640 | 5 | IC50 | = | 3000 | nM | ALA4704018 | 5.52 | nM | Mus musculus | ||
15. | ALA4580568 | 24 | IC50 | = | 81 | nM | ALA4704018 | 7.09 | nM | Mus musculus | ||
16. | ALA4461925 | 30 | IC50 | = | 30 | nM | ALA4704018 | 7.52 | nM | Mus musculus | ||
17. | ALA4640857 | 11; OAT-1441 | IC50 | = | 59 | nM | ALA4704018 | 7.23 | nM | Mus musculus | ||
18. | ALA4206372 | 9 | IC50 | = | 4170 | nM | ALA4704018 | 5.38 | nM | Mus musculus | ||
19. | 1-(3-amino-1H-1,2,4-triazol-5-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | 7f | IC50 | = | 18.8 | nM | ALA4704018 | 7.73 | nM | Mus musculus | ||
20. | 1-(3-amino-1H-1,2,4-triazol-5-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | 7f | Ki | = | 10.5 | nM | ALA4022944 | 7.98 | nM | Mus musculus |