# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5202967 | KPH2f | IC50 | = | 9.37 | uM | ALA5157462 | 5.03 | nM | Homo sapiens | ||
2. | ALA5170470 | Verinurad | INH | 0 | ALA5157444 | NA | % | Homo sapiens | ||||
3. | ALA5178161 | SG1c | INH | = | 15.23 | % | ALA5157444 | % | Homo sapiens | |||
4. | ALA5202967 | KPH2f | INH | = | 50.97 | % | ALA5157444 | % | Homo sapiens | |||
5. | ALA5190525 | KPH1i | INH | = | 23.15 | % | ALA5157444 | % | Homo sapiens | |||
6. | ALA4740905 | 84 | IC50 | = | 32.2 | uM | ALA4670649 | 4.49 | nM | Homo sapiens | ||
7. | ALA4756866 | 83 | IC50 | = | 31.73 | uM | ALA4670649 | 4.50 | nM | Homo sapiens | ||
8. | ALA5284974 | 10 | IC50 | = | 55.96 | uM | ALA5248753 | 4.25 | nM | Homo sapiens | ||
9. | Lesinurad | LESINURAD | INH | 0 | ALA5248752 | Not Active | % | Homo sapiens | ||||
10. | Uric acid | Urate | EC50 | 0 | ALA5209626 | Ec50 Cannot Be Calculated For Isoform 2 | Homo sapiens | |||||
11. | Uric acid | Urate | EC50 | = | 0.3 | mM | ALA5209625 | Substrate (Isoform 1 Only) | nM | Homo sapiens | ||
12. | Orotic acid | SID17388814 | EC50 | = | 1 | mM | ALA5209626 | Substrate | nM | Homo sapiens | ||
13. | Orotic acid | SID17388814 | EC50 | = | 1 | mM | ALA5209625 | Substrate | nM | Homo sapiens | ||
14. | (5Z)-5-[[4-hydroxy-3-(trifluoromethyl)phenyl]methylidene]-3-[4,4,4-trifluoro-2-methyl-2-(2,2,2-trifluoroethyl)butyl]-1,3-thiazolidine-2,4-dione | 30 | INH | = | 34 | % | ALA2061376 | % | Homo sapiens | |||
15. | ALA2057965 | 5 | INH | = | 26 | % | ALA2061376 | % | Homo sapiens |