# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4642294 | Table 2, R9C4 | Activity | = | 60 | % | ALA5244584 | % | Mus musculus | |||
2. | ALA4208325 | 27 | EC50 | = | 193 | nM | ALA4188792 | 6.71 | nM | Mus musculus | ||
3. | GSK137647A | 8, GSK137647A | Rmax | = | 100 | % | ALA3364896 | % | Mus musculus | |||
4. | GSK137647A | 8, GSK137647A | Activity | 0 | ALA3362267 | Not Active | Mus musculus | |||||
5. | GSK137647A | 8, GSK137647A | Activity | 0 | ALA3362266 | Dose-dependent effect | Mus musculus | |||||
6. | AH-7614 | 39 | pIC50 | = | 8.1 | ALA3365231 | 8.10 | nM | Mus musculus | |||
7. | GSK137647A | 8, GSK137647A | pEC50 | = | 6.2 | ALA3364895 | 6.20 | nM | Mus musculus | |||
8. | GSK137647A | 8, GSK137647A | pEC50 | = | 5.2 | ALA3362270 | 5.20 | nM | Mus musculus | |||
9. | ALA4065397 | 29 | %max | = | 108 | % | ALA3996992 | % | Mus musculus | |||
10. | ALA4065397 | 29 | EC50 | = | 70 | nM | ALA3996993 | 7.16 | nM | Mus musculus | ||
11. | ALA3954140 | 22 | EC50 | = | 1300 | nM | ALA3874984 | 5.89 | nM | Mus musculus | ||
12. | ALA3953289 | 21 | EC50 | = | 44 | nM | ALA3874984 | 7.36 | nM | Mus musculus | ||
13. | ALA3893026 | 20 | EC50 | = | 51 | nM | ALA3874984 | 7.29 | nM | Mus musculus | ||
14. | ALA3937916 | 19 | EC50 | = | 670 | nM | ALA3874984 | 6.17 | nM | Mus musculus | ||
15. | ALA3901994 | 18 | EC50 | = | 190 | nM | ALA3874984 | 6.72 | nM | Mus musculus | ||
16. | ALA3973034 | 17 | EC50 | = | 66 | nM | ALA3874984 | 7.18 | nM | Mus musculus | ||
17. | ALA3920891 | 16 | EC50 | > | 10000 | nM | ALA3874984 | nM | Mus musculus | |||
18. | ALA3947837 | 15 | EC50 | = | 590 | nM | ALA3874984 | 6.23 | nM | Mus musculus | ||
19. | 2-[3-[2-chloro-5-(trifluoromethoxy)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid | 14 | EC50 | = | 33 | nM | ALA3874984 | 7.48 | nM | Mus musculus | ||
20. | ALA3891920 | 13 | EC50 | = | 49 | nM | ALA3874984 | 7.31 | nM | Mus musculus |