# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4642294 | Table 2, R9C4 | Activity | = | 60 | % | ALA5244584 | % | Mus musculus | |||
2. | GSK137647A | 8, GSK137647A | Rmax | = | 100 | % | ALA3364896 | % | Mus musculus | |||
3. | GSK137647A | 8, GSK137647A | Activity | 0 | ALA3362267 | Not Active | Mus musculus | |||||
4. | GSK137647A | 8, GSK137647A | Activity | 0 | ALA3362266 | Dose-dependent effect | Mus musculus | |||||
5. | AH-7614 | 39 | pIC50 | = | 8.1 | ALA3365231 | 8.10 | nM | Mus musculus | |||
6. | GSK137647A | 8, GSK137647A | pEC50 | = | 6.2 | ALA3364895 | 6.20 | nM | Mus musculus | |||
7. | GSK137647A | 8, GSK137647A | pEC50 | = | 5.2 | ALA3362270 | 5.20 | nM | Mus musculus | |||
8. | ALA4208325 | 27 | EC50 | = | 193 | nM | ALA4188792 | 6.71 | nM | Mus musculus | ||
9. | ALA4171724 | 4y | EC50 | = | 102 | nM | ALA4134145 | 6.99 | nM | Mus musculus | ||
10. | ALA4165366 | 4x | EC50 | = | 77 | nM | ALA4134145 | 7.11 | nM | Mus musculus | ||
11. | ALA4096579 | 35 | Efficacy | = | 176 | % | ALA4051332 | % | Mus musculus | |||
12. | ALA4078553 | 34 | Efficacy | = | 91 | % | ALA4051332 | % | Mus musculus | |||
13. | ALA4070359 | 33 | Efficacy | = | 79 | % | ALA4051332 | % | Mus musculus | |||
14. | ALA4097537 | 32 | Efficacy | = | 99 | % | ALA4051332 | % | Mus musculus | |||
15. | ALA4080998 | 31 | Efficacy | = | 103 | % | ALA4051332 | % | Mus musculus | |||
16. | ALA4105241 | 30 | Efficacy | = | 112 | % | ALA4051332 | % | Mus musculus | |||
17. | ALA4102951 | 29 | Efficacy | = | 99 | % | ALA4051332 | % | Mus musculus | |||
18. | ALA4096579 | 35 | EC50 | = | 0.017 | uM | ALA4051331 | 7.77 | nM | Mus musculus | ||
19. | ALA4078553 | 34 | EC50 | = | 0.51 | uM | ALA4051331 | 6.29 | nM | Mus musculus | ||
20. | ALA4070359 | 33 | EC50 | = | 1 | uM | ALA4051331 | 6.00 | nM | Mus musculus |