# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Nrf2 peptide | AFFAQLQLDEETGEFL | IC50 | = | 33 | nM | ALA2406877 | 7.48 | nM | Homo sapiens | ||
2. | ALA2402206 | 15 | IC50 | = | 118 | uM | ALA2406877 | nM | Homo sapiens | |||
3. | ALA2402207 | 16 | IC50 | = | 2.7 | uM | ALA2406877 | 5.57 | nM | Homo sapiens | ||
4. | ALA2402207 | 16 | Activity | 0 | ALA2406876 | Not Active | Homo sapiens | |||||
5. | Dimethyl fumarate | DIMETHYL FUMARATE | Activity | 0 | ALA2406876 | Active | Homo sapiens | |||||
6. | ALA2402206 | 15 | Activity | 0 | ALA2406872 | Active | Homo sapiens | |||||
7. | ALA2402207 | 16 | Activity | 0 | ALA2406872 | Active | Homo sapiens | |||||
8. | ALA1460757 | SID864554 | Kd | = | 1.9 | uM | ALA2382890 | 5.72 | nM | Homo sapiens | ||
9. | ML 334 | (SRS)-5, ML334, LH601A, isomer A, | Kd | = | 1 | uM | ALA2382890 | 6.00 | nM | Homo sapiens | ||
10. | ALA2381969 | (RSR)-5, isomer B | Kd | = | 100 | uM | ALA2382890 | 4.00 | nM | Homo sapiens | ||
11. | ALA2381970 | (SSR/RRS)-5, diastereomer C/D | Kd | = | 700 | uM | ALA2382890 | nM | Homo sapiens | |||
12. | ALA2381966 | (SRR)-5 | Activity | 0 | ALA2382890 | Not Active | Homo sapiens | |||||
13. | ALA2381964 | (RSS)-5 | Activity | 0 | ALA2382890 | Not Active | Homo sapiens | |||||
14. | ALA2381967 | (SSS)-5 | Activity | 0 | ALA2382890 | Not Active | Homo sapiens | |||||
15. | ALA2381965 | (RRR)-5 | Activity | 0 | ALA2382890 | Not Active | Homo sapiens | |||||
16. | ALA1502018 | SID49679494 | Max_Activity_Concent | 50 | uM | ALA2114882 | active | uM | Homo sapiens | |||
17. | ALA1423626 | SID26542735 | Max_Activity_Concent | 0.8 | uM | ALA2114882 | inactive | uM | Homo sapiens | |||
18. | ALA1370910 | SID49646559 | Max_Activity_Concent | 0.38 | uM | ALA2114882 | inactive | uM | Homo sapiens | |||
19. | ALA1420227 | SID49821344 | Max_Activity_Concent | 0.8 | uM | ALA2114882 | inactive | uM | Homo sapiens | |||
20. | ALA1566994 | SID24780599 | Max_Activity_Concent | 50 | uM | ALA2114882 | active | uM | Homo sapiens |