# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405591 | % | Homo sapiens | |||
2. | BI 605906 | BI605906 | % Ctrl | 90 | % | ALA4887329 | Not Active | % | Homo sapiens | |||
3. | ALA4097778 | 16h | pIC50 | 6 | ALA4885453 | nM | Homo sapiens | |||||
4. | ALA4549667 | EUB0000720 | pIC50 | 6 | ALA4885169 | nM | Homo sapiens | |||||
5. | ALA4088216 | 14 | pIC50 | 6 | ALA4884878 | nM | Homo sapiens | |||||
6. | Tivantinib (ARQ 197) | TIVANTINIB | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
7. | Tirbanibulin | 3, KX-01 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
8. | K-252a | 2 (K-252a) | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
9. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
10. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
11. | Alisertib (MLN8237) | 9, MLN-8237 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
12. | Trametinib (GSK1120212) | TRAMETINIB | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
13. | Nilotinib (AMN-107) | 38 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
14. | ridaforolimus | RIDAFOROLIMUS | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
15. | HMN-214 | HMN-214 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
16. | Gedatolisib (PF-05212384, PKI-587) | 26, PKI-587 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
17. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
18. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
19. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens | ||
20. | GSK461364 | GSK-461364A | Kd apparent | > | 30000 | nM | ALA3991908 | Inactive | nM | Homo sapiens |