# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Cimetidine | cimetidine | IC50 | = | 8 | uM | ALA2077062 | 5.10 | inhibitor [IC50=8uM] | nM | Mus musculus | |
2. | 4-Amino-N-(2-diethylaminoethyl)benzamide | Procainamide | IC50 | = | 312 | uM | ALA2077062 | inhibitor [IC50=312uM] | nM | Mus musculus | ||
3. | tetraethylammonium | 1 | IC50 | = | 3.5 | uM | ALA2077062 | 5.46 | inhibitor [IC50=3.5uM] | nM | Mus musculus | |
4. | Choline | Choline | IC50 | = | 217 | uM | ALA2077062 | inhibitor [IC50=217uM] | nM | Mus musculus | ||
5. | Quinine | 10a | IC50 | = | 2.8 | uM | ALA2077062 | 5.55 | inhibitor [IC50=2.8uM] | nM | Mus musculus | |
6. | N-Methylnicotinamide | 15 | IC50 | = | 13661 | uM | ALA2077062 | inhibitor [IC50=13661uM] | nM | Mus musculus | ||
7. | tetraethylammonium | 1 | Km | = | 35.7 | uM | ALA2075959 | substrate [Km=35.7uM] | nM | Mus musculus | ||
8. | MPP⁺ | 1 | Km | = | 24 | uM | ALA2075959 | substrate [Km=24uM] | nM | Mus musculus |