# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-[2-[5-chloro-2-[(5-ethoxyquinolin-8-yl)sulfonylamino]phenyl]ethynyl]-4-methoxypyridine-2-carboxylic acid | EUB0001566 | IC50 | = | 638 | uM | ALA5242471 | nM | Homo sapiens | |||
2. | 5-[2-[5-chloro-2-[(5-ethoxyquinolin-8-yl)sulfonylamino]phenyl]ethynyl]-4-methoxypyridine-2-carboxylic acid | EUB0001566 | IC50 | > | 25000 | uM | ALA5242470 | nM | Homo sapiens | |||
3. | ALA5276884 | 18k | IC50 | = | 239 | nM | ALA5242457 | 6.62 | nM | Homo sapiens | ||
4. | ALA5276884 | 18k | IC50 | = | 137 | nM | ALA5242456 | 6.86 | nM | Homo sapiens | ||
5. | 5-[2-[5-chloro-2-[(5-ethoxyquinolin-8-yl)sulfonylamino]phenyl]ethynyl]-4-methoxypyridine-2-carboxylic acid | EUB0001566 | IC50 | > | 4 | uM | ALA5242455 | nM | Homo sapiens | |||
6. | AR-C155858 | 13 | IC50 | = | 6.2 | nM | ALA5242455 | 8.21 | nM | Homo sapiens | ||
7. | ALA3335793 | 39, AZD3965 | IC50 | = | 22 | nM | ALA5242455 | 7.66 | nM | Homo sapiens | ||
8. | ALA5287835 | 17l | IC50 | > | 50000 | nM | ALA5242455 | nM | Homo sapiens | |||
9. | ALA5282741 | 18j | IC50 | = | 10000 | nM | ALA5242455 | 5.00 | nM | Homo sapiens | ||
10. | ALA5267752 | 18h | IC50 | > | 50000 | nM | ALA5242455 | nM | Homo sapiens | |||
11. | AR-C155858 | 13 | IC50 | = | 2.5 | nM | ALA5242454 | 8.60 | nM | Homo sapiens | ||
12. | ALA3335793 | 39, AZD3965 | IC50 | = | 7.1 | nM | ALA5242454 | 8.15 | nM | Homo sapiens | ||
13. | ALA5287835 | 17l | IC50 | = | 2700 | nM | ALA5242454 | 5.57 | nM | Homo sapiens | ||
14. | ALA5282741 | 18j | IC50 | = | 8200 | nM | ALA5242454 | 5.09 | nM | Homo sapiens | ||
15. | ALA5267752 | 18h | IC50 | = | 13000 | nM | ALA5242454 | 4.89 | nM | Homo sapiens | ||
16. | AR-C155858 | 13 | IC50 | > | 30000 | nM | ALA5242453 | nM | Homo sapiens | |||
17. | ALA3335793 | 39, AZD3965 | IC50 | > | 30000 | nM | ALA5242453 | nM | Homo sapiens | |||
18. | ALA5287835 | 17l | IC50 | = | 21 | nM | ALA5242453 | 7.68 | nM | Homo sapiens | ||
19. | ALA5282741 | 18j | IC50 | = | 13 | nM | ALA5242453 | 7.89 | nM | Homo sapiens | ||
20. | ALA5267752 | 18h | IC50 | = | 18 | nM | ALA5242453 | 7.75 | nM | Homo sapiens |