| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1236196 | Tetrabuthylammonium | Ki | = | 7.3 | uM | ALA2077854 | 5.14 | inhibitor [Ki=7.3uM] | nM | Mus musculus | |
| 2. |  ALA1209651 | 28 | Ki | = | 2040 | uM | ALA2077854 | inhibitor [Ki=2040uM] | nM | Mus musculus | ||
| 3. |  ALA2074857 | Tetrapropylammonium | Ki | = | 19.8 | uM | ALA2077854 | 4.70 | inhibitor [Ki=19.8uM] | nM | Mus musculus | |
| 4. |  tetraethylammonium | 1 | Ki | = | 128 | uM | ALA2077854 | inhibitor [Ki=128uM] | nM | Mus musculus | ||
| 5. |  Choline | Choline | Activity | 0 | ALA2077909 | is not a substrate [-] | Mus musculus | |||||
| 6. |  Cimetidine | cimetidine | Activity | 0 | ALA2077909 | is not a substrate [-] | Mus musculus | |||||
| 7. |  N-Methylnicotinamide | 15 | IC50 | = | 7337 | uM | ALA2077071 | inhibitor [IC50=7337uM] | nM | Mus musculus | ||
| 8. | Choline | Choline | IC50 | = | 55 | uM | ALA2077071 | 4.26 | inhibitor [IC50=55uM] | nM | Mus musculus | |
| 9. |  4-Amino-N-(2-diethylaminoethyl)benzamide | Procainamide | IC50 | = | 3.9 | uM | ALA2077071 | 5.41 | inhibitor [IC50=3.9uM] | nM | Mus musculus | |
| 10. |  ALA2074704 | Tetrapentylammonium | Activity | 0 | ALA2077816 | inhibitor [trans-inhibited: (at a rough estimate) 30 % of control] | Mus musculus | |||||
| 11. | Cimetidine | cimetidine | IC50 | = | 0.59 | uM | ALA2077071 | 6.23 | inhibitor [IC50=0.59uM] | nM | Mus musculus | |
| 12. | tetraethylammonium | 1 | IC50 | = | 0.54 | uM | ALA2077071 | 6.27 | inhibitor [IC50=0.54uM] | nM | Mus musculus | |
| 13. |  Quinine | 10a | IC50 | = | 0.28 | uM | ALA2077071 | 6.55 | inhibitor [IC50=0.28uM] | nM | Mus musculus | |
| 14. | ALA1236196 | Tetrabuthylammonium | Km | = | 43 | uM | ALA2075998 | substrate [Km=43uM] | nM | Mus musculus | ||
| 15. | Choline | Choline | Km | = | 42 | uM | ALA2075998 | substrate [Km=42uM] | nM | Mus musculus | ||
| 16. | tetraethylammonium | 1 | Km | = | 38 | uM | ALA2075997 | substrate [Km=38uM] | nM | Mus musculus | ||
| 17. |  [³H]thiamine | 1, thiamine | Activity | = | 12.7 | % | ALA2077821 | inhibitor [12.7 % of control] | % | Mus musculus | ||
| 18. | ALA1209651 | 28 | Activity | = | 0 | % | ALA2077818 | inhibitor [0 % of control] | % | Mus musculus | ||
| 19. | [³H]thiamine | 1, thiamine | Activity | = | 0 | % | ALA2077817 | inhibitor [0 % of control] | % | Mus musculus | ||
| 20. |  Quinidine | quinidine | Activity | = | 0 | % | ALA2077819 | inhibitor [0 % of control] | % | Mus musculus |
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