| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Cefadroxil | 85(Cefadroxil) | IC50 | = | 1780 | uM | ALA3537401 | nM | Rattus norvegicus | |||
| 2. |  ALA4105032 | 10; PF-06679142 | Ratio | = | 2.3 | ALA4023969 | Rattus norvegicus | |||||
| 3. |  ALA3986871 | BDBM238079 | Ratio | = | 2 | ALA4023969 | Rattus norvegicus | |||||
| 4. |  PF 06409577 | 7 | Ratio | = | 8.3 | ALA4023969 | Rattus norvegicus | |||||
| 5. |  [³H]taurocholic acid | THCA | Activity | 0 | ALA2078239 | inhibitor [(at a rough estimate) 50 % of control] | Rattus norvegicus | |||||
| 6. |  [³H]BSP | Bromosulfophthalein | Activity | 0 | ALA2078254 | inhibitor [(at a rough estimate) 5 % of control] | Rattus norvegicus | |||||
| 7. |  Cefoperazone | Cefoperazone | Activity | 0 | ALA2078251 | inhibitor [(at a rough estimate) 40 % of control] | Rattus norvegicus | |||||
| 8. | [³H]taurocholic acid | THCA | Activity | 0 | ALA2078252 | inhibitor [(at a rough estimate) 35 % of control] | Rattus norvegicus | |||||
| 9. |  [³H]methotrexate | 138 | Activity | 0 | ALA2078245 | inhibitor [(at a rough estimate) 35 % of control] | Rattus norvegicus | |||||
| 10. |  estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Ki | = | 9.1 | uM | ALA2075297 | 5.04 | inhibitor [Ki=9.1uM] | nM | Rattus norvegicus | |
| 11. | [³H]taurocholic acid | THCA | Ki | = | 790 | uM | ALA2076869 | inhibitor [Ki=790uM] | nM | Rattus norvegicus | ||
| 12. |  Cefazolin | 19 | Ki | = | 780 | uM | ALA2076054 | inhibitor [Ki=780uM] | nM | Rattus norvegicus | ||
| 13. | Cefoperazone | Cefoperazone | Ki | = | 670 | uM | ALA2076054 | inhibitor [Ki=670uM] | nM | Rattus norvegicus | ||
| 14. |  Indoxyl acetate | Indole acetate | Ki | = | 582 | uM | ALA2075296 | inhibitor [Ki=582uM] | nM | Rattus norvegicus | ||
| 15. |  penicillin G | Benzylpenicillin | Ki | = | 52.8 | uM | ALA2076478 | 4.28 | inhibitor [Ki=52.8uM] | nM | Rattus norvegicus | |
| 16. |  Cephalothin | Cephalothin | Ki | = | 48 | uM | ALA2076054 | 4.32 | inhibitor [Ki=48uM] | nM | Rattus norvegicus | |
| 17. |  Cimetidine | cimetidine | Ki | = | 46.8 | uM | ALA2075297 | 4.33 | inhibitor [Ki=46.8uM] | nM | Rattus norvegicus | |
| 18. |  Probenecid | probenecid | Ki | = | 4.43 | uM | ALA2076479 | 5.35 | inhibitor [Ki=4.43uM] | nM | Rattus norvegicus | |
| 19. |  4-Aminohippuric Acid | 6d | Ki | = | 398 | uM | ALA2076479 | inhibitor [Ki=398uM] | nM | Rattus norvegicus | ||
| 20. |  [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Ki | = | 35.6 | uM | ALA2076479 | 4.45 | inhibitor [Ki=35.6uM] | nM | Rattus norvegicus |
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