# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 4-Amino-N-(2-diethylaminoethyl)benzamide | Procainamide | IC50 | = | 1 | mM | ALA2077083 | inhibitor [IC501mM] | nM | Rattus norvegicus | ||
2. | tetraethylammonium | 1 | IC50 | = | 1 | mM | ALA2077083 | inhibitor [IC501mM] | nM | Rattus norvegicus | ||
3. | Cimetidine | cimetidine | IC50 | = | 1.5 | mM | ALA2077083 | inhibitor [IC501.5mM] | nM | Rattus norvegicus | ||
4. | 5-(N,N-Dimethyl)amiloride hydrochloride | 5h | IC50 | = | 0.2 | mM | ALA2077083 | inhibitor [IC500.2mM] | nM | Rattus norvegicus | ||
5. | desipramine | desmethylimipramine | IC50 | = | 0.08 | mM | ALA2077083 | 4.10 | inhibitor [IC500.08mM] | nM | Rattus norvegicus | |
6. | Amiloride | 1 | Activity | = | 79 | % | ALA2078260 | inhibitor [79% of control] | % | Rattus norvegicus | ||
7. | tetraethylammonium | 1 | Activity | 0 | ALA2078256 | substrate [IC50] | Rattus norvegicus | |||||
8. | ALA3 | 2 | Activity | = | 29 | % | ALA2078258 | inhibitor [29% of control] | % | Rattus norvegicus | ||
9. | Verapamil | 24 | Activity | = | 20 | % | ALA2078257 | inhibitor [20% of control] | % | Rattus norvegicus | ||
10. | MPP⁺ | 1 | Activity | = | 62 | % | ALA2078585 | inhibitor [62% of control] | % | Rattus norvegicus | ||
11. | Imipramine | Imipramine | Activity | = | 31 | % | ALA2078259 | inhibitor [31% of control] | % | Rattus norvegicus |