# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | L-(+)-Ergothioneine | L-Ergothioneine | EC50 | = | 40 | uM | ALA5209595 | 4.40 | Substrate | nM | Homo sapiens | |
2. | Quinidine | quinidine | INH | = | 83.9 | % | ALA3531371 | % | Homo sapiens | |||
3. | Linagliptin | 1, BI 1356 | INH | = | 19.4 | % | ALA3531367 | % | Homo sapiens | |||
4. | Linagliptin | 1, BI 1356 | Drug uptake | 0 | ALA3536918 | Not Active | Homo sapiens | |||||
5. | L-Lysine | L-Lysine | Activity | 0 | ALA2076162 | is not an inhibitor [-] | Homo sapiens | |||||
6. | N-Methylnicotinamide | 15 | Activity | 0 | ALA2076161 | is not an inhibitor [-] | Homo sapiens | |||||
7. | 4-Aminohippuric Acid | 6d | Activity | 0 | ALA2076158 | is not an inhibitor [-] | Homo sapiens | |||||
8. | penicillin G | Benzylpenicillin | Activity | 0 | ALA2077088 | is not a substrate [-] | Homo sapiens | |||||
9. | penicillin G | Benzylpenicillin | Activity | 0 | ALA2076157 | is not an inhibitor [-] | Homo sapiens | |||||
10. | 1,4-Diaminobutane | Putrescine | Activity | 0 | ALA2076155 | is not an inhibitor [-] | Homo sapiens | |||||
11. | Spermidine | spermidine | Activity | 0 | ALA2076151 | is not an inhibitor [-] | Homo sapiens | |||||
12. | Spermine | spermine | Activity | 0 | ALA2076017 | is not an inhibitor [-] | Homo sapiens | |||||
13. | L-Arginine | 35 | Activity | 0 | ALA2076170 | is not an inhibitor [-] | Homo sapiens | |||||
14. | tetraethylammonium | 1 | Km | = | 436 | uM | ALA2076015 | substrate [Km=436uM] | nM | Homo sapiens | ||
15. | guanidine | 14 | Activity | = | 89.6 | % | ALA2077910 | inhibitor [89.6 % of control] | % | Homo sapiens | ||
16. | Verapamil | 24 | Activity | = | 8.8 | % | ALA2076016 | inhibitor [8.8 % of control] | % | Homo sapiens | ||
17. | clonidine | clonidine | Activity | = | 70.9 | % | ALA2076166 | inhibitor [70.9 % of control] | % | Homo sapiens | ||
18. | DL-Carnitine | Carnitine | Activity | 0 | ALA2077088 | substrate [+] | Homo sapiens | |||||
19. | mepyramine | Mepyramine | Activity | 0 | ALA2077088 | substrate [+] | Homo sapiens | |||||
20. | Quinidine | quinidine | Activity | 0 | ALA2077088 | substrate [+] | Homo sapiens |