| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  [³H]taurocholic acid | THCA | Activity | 0 | ALA2077034 | inhibitor [(at a rough estimate) 55 % of control] | Rattus norvegicus | |||||
| 2. |  Rifampicin | rifampacin | Activity | 0 | ALA2077029 | inhibitor [(at a rough estimate) 15 % of control] | Rattus norvegicus | |||||
| 3. |  Cefoperazone | Cefoperazone | Activity | 0 | ALA2077033 | inhibitor [(at a rough estimate) 15 % of control] | Rattus norvegicus | |||||
| 4. |  4-[(2Z)-2-[(2E,4E,6Z)-7-[1,1-dimethyl-3-(4-sulfobutyl)benzo[e]indol-3-ium-2-yl]hepta-2,4,6-trienylidene]-1,1-dimethylbenzo[e]indol-3-yl]butane-1-sulfonate | SID50125759 | Activity | 0 | ALA2077031 | inhibitor [(at a rough estimate) 10 % of control] | Rattus norvegicus | |||||
| 5. |  Bumetanide | 160 | Activity | 0 | ALA2077035 | inhibitor [(at a rough estimate) 10 % of control] | Rattus norvegicus | |||||
| 6. |  Bromosulfalein | Bromosulfophthalein | Activity | 0 | ALA2077036 | inhibitor [(at a rough estimate) <5 % of control] | Rattus norvegicus | |||||
| 7. |  Ketoprofen | ketoprofen | Activity | 0 | ALA2077030 | inhibitor [(at a rough estimate) <0 % of control] | Rattus norvegicus | |||||
| 8. |  tetraethylammonium | 1 | Activity | 0 | ALA2078540 | is not a substrate [-] | Rattus norvegicus | |||||
| 9. |  Glyburide | 2 | Ki | = | 12.3 | uM | ALA2077860 | 4.91 | inhibitor [Ki=12.3uM] | nM | Rattus norvegicus | |
| 10. | Ketoprofen | ketoprofen | Ki | = | 1.84 | uM | ALA2077860 | 5.74 | inhibitor [Ki=1.84uM] | nM | Rattus norvegicus | |
| 11. | 4-[(2Z)-2-[(2E,4E,6Z)-7-[1,1-dimethyl-3-(4-sulfobutyl)benzo[e]indol-3-ium-2-yl]hepta-2,4,6-trienylidene]-1,1-dimethylbenzo[e]indol-3-yl]butane-1-sulfonate | SID50125759 | Ki | = | 1.15 | uM | ALA2077860 | 5.94 | inhibitor [Ki=1.15uM] | nM | Rattus norvegicus | |
| 12. |  Probenecid | probenecid | IC50 | = | 977 | uM | ALA2075807 | inhibitor [IC50=977 +/- 265uM] | nM | Rattus norvegicus | ||
| 13. |  Pravastatin | 2 (pravastatin) | IC50 | = | 449 | uM | ALA2075807 | inhibitor [IC50=449 +/- 105uM] | nM | Rattus norvegicus | ||
| 14. |  Testosterone | 21 | Activity | 0 | ALA2077037 | inducer [Decrease] | Rattus norvegicus | |||||
| 15. |  Salicylic acid | 17 | Km | = | 88.8 | uM | ALA2078540 | substrate [Km=88.8uM] | nM | Rattus norvegicus | ||
| 16. | Salicylic acid | 17 | Km | = | 81.2 | uM | ALA2077095 | substrate [Km=81.2uM] | nM | Rattus norvegicus | ||
| 17. |  Prostaglandin E₂ | PGE2 | Km | = | 38.5 | uM | ALA2077095 | substrate [Km=38.5uM] | nM | Rattus norvegicus | ||
| 18. |  Dinoprost | 9 | Km | = | 414 | nM | ALA2077028 | substrate [Km414nM] | nM | Rattus norvegicus | ||
| 19. |  cefamandole | cefamandol | IC50 | = | 3.18 | mM | ALA2077096 | inhibitor [IC503.18mM] | nM | Rattus norvegicus | ||
| 20. | Cefoperazone | Cefoperazone | IC50 | = | 1.62 | mM | ALA2077096 | inhibitor [IC501.62mM] | nM | Rattus norvegicus |
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