| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Cimetidine | cimetidine | Activity | 0 | ALA2078183 | inhibitor [(at a rough estimate) 30 % of control] | Homo sapiens | |||||
| 2. |  4-Amino-N-(2-diethylaminoethyl)benzamide | Procainamide | Ki | = | 738 | uM | ALA2078549 | inhibitor [Ki=738uM] | nM | Homo sapiens | ||
| 3. |  guanidine | 14 | Ki | = | 6201 | uM | ALA2078549 | inhibitor [Ki=6201uM] | nM | Homo sapiens | ||
| 4. |  MPP⁺ | 1 | Ki | = | 54 | uM | ALA2078549 | 4.27 | inhibitor [Ki=54uM] | nM | Homo sapiens | |
| 5. |  Imipramine | Imipramine | Ki | = | 42 | uM | ALA2078549 | 4.38 | inhibitor [Ki=42uM] | nM | Homo sapiens | |
| 6. |  clonidine | clonidine | Ki | = | 373 | uM | ALA2078549 | inhibitor [Ki=373uM] | nM | Homo sapiens | ||
| 7. |  desipramine | desmethylimipramine | Ki | = | 14 | uM | ALA2078549 | 4.85 | inhibitor [Ki=14uM] | nM | Homo sapiens | |
| 8. |  Histamine, Free Base | histamine | Ki | = | 140 | uM | ALA2078182 | inhibitor [Ki=140uM] | nM | Homo sapiens | ||
| 9. |  tetraethylammonium | 1 | Ki | = | 1372 | uM | ALA2078549 | inhibitor [Ki=1372uM] | nM | Homo sapiens | ||
| 10. |  Colchicine | colchicine | Ki | = | 0.12 | uM | ALA2075864 | 6.92 | inhibitor [Ki=0.12uM] | nM | Homo sapiens | |
| 11. |  disprocynium24 | 1d | Ki | = | 0.015 | uM | ALA2075864 | 7.82 | inhibitor [Ki=0.015uM] | nM | Homo sapiens | |
| 12. | clonidine | clonidine | IC50 | = | 79.3 | uM | ALA2077362 | 4.10 | inhibitor [IC50=79.3uM] | nM | Homo sapiens | |
| 13. |  phenoxybenzamine | Phenoxybenzamine | IC50 | = | 6.13 | uM | ALA2077954 | 5.21 | inhibitor [IC50=6.13uM] | nM | Homo sapiens | |
| 14. |  ALA2074647 | o-Methylisoprenaline | IC50 | = | 4.38 | uM | ALA2077954 | 5.36 | inhibitor [IC50=4.38uM] | nM | Homo sapiens | |
| 15. |  ALA103 | Progesterone | IC50 | = | 4.28 | uM | ALA2077954 | 5.37 | inhibitor [IC50=4.28uM] | nM | Homo sapiens | |
| 16. |  β-Estradiol | Table II | IC50 | = | 2.88 | uM | ALA2077954 | 5.54 | inhibitor [IC50=2.88uM] | nM | Homo sapiens | |
| 17. |  [³H]prazosin | 1 | IC50 | = | 12.6 | uM | ALA2077954 | 4.90 | inhibitor [IC50=12.6uM] | nM | Homo sapiens | |
| 18. | tetraethylammonium | 1 | IC50 | = | 10300 | uM | ALA2077362 | inhibitor [IC50=10300uM] | nM | Homo sapiens | ||
| 19. |  ALA2074851 | Cyanine-863 | IC50 | = | 1.76 | uM | ALA2077362 | 5.75 | inhibitor [IC50=1.76uM] | nM | Homo sapiens | |
| 20. |  Corticosterone | 7 | IC50 | = | 0.29 | uM | ALA2077954 | 6.54 | inhibitor [IC50=0.29uM] | nM | Homo sapiens |
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