| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2074926 | Tauroallocholate | Activity | 0 | ALA2078225 | inhibitor [(at a rough estimate) 50 % of control] | Rattus norvegicus | |||||
| 2. |  ALA2074708 | Bosentan M2 | Ki | = | 8.5 | uM | ALA2075960 | 5.07 | inhibitor [Ki=8.5uM] | nM | Rattus norvegicus | |
| 3. |  Glyburide | 2 | Ki | = | 6.1 | uM | ALA2076297 | 5.21 | inhibitor [Ki=6.1uM] | nM | Rattus norvegicus | |
| 4. |  rifamycin SV | 1b(rifamycin SV) | Ki | = | 3.8 | uM | ALA2076297 | 5.42 | inhibitor [Ki=3.8uM] | nM | Rattus norvegicus | |
| 5. |  Fusidic Acid | Fusidic acid | Ki | = | 2.2 | uM | ALA2078221 | 5.66 | inhibitor [Ki=2.2uM] | nM | Rattus norvegicus | |
| 6. |  Bosentan | Bosentan | Ki | = | 12 | uM | ALA2075960 | 4.92 | inhibitor [Ki=12uM] | nM | Rattus norvegicus | |
| 7. |  Rifampicin | rifampacin | Ki | = | 11.9 | uM | ALA2076297 | 4.92 | inhibitor [Ki=11.9uM] | nM | Rattus norvegicus | |
| 8. |  Cyclosporin A | 1a Cys-A | Ki | = | 0.3 | uM | ALA2076297 | 6.52 | inhibitor [Ki=0.3uM] | nM | Rattus norvegicus | |
| 9. | ALA2074926 | Tauroallocholate | Activity | 0 | ALA2078219 | is not a substrate [-] | Rattus norvegicus | |||||
| 10. |  [³H]taurocholic acid | THCA | Activity | 0 | ALA2078217 | is not a substrate [-] | Rattus norvegicus | |||||
| 11. | Glyburide | 2 | IC50 | = | 8.6 | uM | ALA2075962 | 5.07 | inhibitor [IC50=8.6uM] | nM | Rattus norvegicus | |
| 12. |  ALA2074736 | Taurochenodeoxycholate sulfate | IC50 | = | 67.9 | uM | ALA2075961 | 4.17 | inhibitor [IC50=67.9uM] | nM | Rattus norvegicus | |
| 13. |  ALA2074644 | Taurolithocholate-3-sulfate | IC50 | = | 61.9 | uM | ALA2075961 | 4.21 | inhibitor [IC50=61.9uM] | nM | Rattus norvegicus | |
| 14. |  Ethinyl Estradiol | 17 alpha-ethynyl E2 | Activity | 0 | ALA2078222 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 15. |  [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Activity | 0 | ALA2078226 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 16. |  β-Sitosterol | 13 | Activity | 0 | ALA2078220 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 17. | ALA2074736 | Taurochenodeoxycholate sulfate | IC50 | = | 4.6 | uM | ALA2075963 | 5.34 | inhibitor [IC50=4.6uM] | nM | Rattus norvegicus | |
| 18. |  ALA408 | Troglitazone | IC50 | = | 3.9 | uM | ALA2077363 | 5.41 | inhibitor [IC50=3.9uM] | nM | Rattus norvegicus | |
| 19. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Activity | 0 | ALA2078277 | inducer [Decrease] | Rattus norvegicus | |||||
| 20. |  ALA3351088 | Endotoxin | Activity | 0 | ALA2078227 | inducer [Decrease] | Rattus norvegicus |
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