| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Lesinurad | LESINURAD | IC50 | = | 2.03 | uM | ALA4357103 | 5.69 | nM | Homo sapiens | ||
| 2. | Lesinurad | LESINURAD | IC50 | = | 7.3 | uM | ALA4610168 | 5.14 | nM | Homo sapiens | ||
| 3. |  Probenecid | probenecid | IC50 | = | 54.9 | uM | ALA4610168 | 4.26 | nM | Homo sapiens | ||
| 4. | Probenecid | probenecid | INH | = | 81.4 | % | ALA3531370 | % | Homo sapiens | |||
| 5. |  Linagliptin | 1, BI 1356 | INH | = | 0 | % | ALA3536929 | % | Homo sapiens | |||
| 6. | Linagliptin | 1, BI 1356 | Drug uptake | 0 | ALA3536914 | Not Active | Homo sapiens | |||||
| 7. |  ALA3929544 | 47 | IC50 | = | 8.5 | uM | ALA3853579 | 5.07 | nM | Homo sapiens | ||
| 8. |  ALA3924161 | 46 | IC50 | = | 9.4 | uM | ALA3853579 | 5.03 | nM | Homo sapiens | ||
| 9. |  ALA3683287 | BDBM165667 | IC50 | = | 14 | uM | ALA3853461 | 4.85 | nM | Homo sapiens | ||
| 10. |  ALA3688197 | BDBM165905 | IC50 | = | 15 | uM | ALA3853461 | 4.82 | nM | Homo sapiens | ||
| 11. |  Indomethacin | Indomethacin | Activity | 0 | ALA2075521 | inhibitor [(at a rough estimate) 5 % of control] | Homo sapiens | |||||
| 12. |  Furosemide | furosemide | Activity | 0 | ALA2075524 | inhibitor [(at a rough estimate) 5 % of control] | Homo sapiens | |||||
| 13. |  Diclofenac | 25 (Diclofenac) | Activity | 0 | ALA2075527 | inhibitor [(at a rough estimate) 5 % of control] | Homo sapiens | |||||
| 14. |  ALA2074784 | 4-methylumbelliferone sulfate | Activity | 0 | ALA2075534 | inhibitor [(at a rough estimate) 40 % of control] | Homo sapiens | |||||
| 15. |  Corticosterone | 7 | Activity | 0 | ALA2075529 | inhibitor [(at a rough estimate) 30 % of control] | Homo sapiens | |||||
| 16. |  Cefotaxime acid | cefotaxime | Ki | = | 6.15 | uM | ALA2078490 | 5.21 | inhibitor [Ki=6.15uM] | nM | Homo sapiens | |
| 17. | Probenecid | probenecid | Ki | = | 54.9 | uM | ALA2076874 | 4.26 | inhibitor [Ki=54.9uM] | nM | Homo sapiens | |
| 18. |  Betamipron | SID26746918 | Ki | = | 502 | uM | ALA2076874 | inhibitor [Ki=502uM] | nM | Homo sapiens | ||
| 19. | Probenecid | probenecid | Ki | = | 44.4 | uM | ALA2077547 | 4.35 | inhibitor [Ki=44.4uM] | nM | Homo sapiens | |
| 20. |  ALA510139 | Citrinin | Ki | = | 366.4 | uM | ALA2077547 | inhibitor [Ki=366.4uM] | nM | Homo sapiens |
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