# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [³H]taurocholic acid | THCA | Activity | 0 | ALA2077130 | inhibitor [(at a rough estimate) 55 % of control] | Homo sapiens | |||||
2. | 3,3',5-Triiodo-L-thyronine | 11 | Activity | 0 | ALA2077128 | inhibitor [(at a rough estimate) 30 % of control] | Homo sapiens | |||||
3. | Bromosulfalein | Bromosulfophthalein | Activity | 0 | ALA2077129 | inhibitor [(at a rough estimate) 15 % of control] | Homo sapiens | |||||
4. | L-Thyroxine | 181 (Thyroxine) | Activity | 0 | ALA2077131 | inhibitor [(at a rough estimate) 15 % of control] | Homo sapiens | |||||
5. | Unoprostone isopropyl ester | UNOPROSTONE ISOPROPYL | Activity | 0 | ALA2077874 | is not a substrate [(-)] | Homo sapiens | |||||
6. | 3,3′,5′-Triiodo-L-thyronine | reverse tri-iodothyronine (r-T3) | Activity | 0 | ALA2077553 | substrate [+] | Homo sapiens | |||||
7. | L-Thyroxine | 181 (Thyroxine) | Activity | 0 | ALA2077553 | substrate [+] | Homo sapiens | |||||
8. | 17β-Estradiol 17β-D-Glucuronide | estradiol 17b glucuronide | Activity | 0 | ALA2077554 | substrate [+] | Homo sapiens | |||||
9. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Activity | 0 | ALA2077554 | substrate [+] | Homo sapiens | |||||
10. | penicillin G | Benzylpenicillin | Activity | 0 | ALA2077554 | substrate [+] | Homo sapiens | |||||
11. | Prostaglandin E₂ | PGE2 | Activity | 0 | ALA2077554 | substrate [+] | Homo sapiens | |||||
12. | [³H]taurocholic acid | THCA | Km | = | 14.9 | uM | ALA2077553 | substrate [Km=14.9uM] | nM | Homo sapiens | ||
13. | Unoprostone | unoprostone | Km | = | 132 | uM | ALA2077874 | substrate [Km=132uM] | nM | Homo sapiens | ||
14. | 3,3',5-Triiodo-L-thyronine | 11 | Km | = | 0.9 | uM | ALA2077553 | substrate [Km=0.9uM] | nM | Homo sapiens |