| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Probenecid | probenecid | Activity | 0 | ALA2078027 | inhibitor [(at a rough estimate) 35 % of control] | Rattus norvegicus | |||||
| 2. |  ALA213947 | M2 | Ki | = | 83.8 | uM | ALA2077359 | 4.08 | inhibitor [Ki=83.8uM] | nM | Rattus norvegicus | |
| 3. |  ALA493586 | 4-methylumbelliferone glucuronide | Ki | = | 77 | uM | ALA2077359 | 4.11 | inhibitor [Ki=77uM] | nM | Rattus norvegicus | |
| 4. |  ALA2074599 | E3040 glucuronide | Ki | = | 2.6 | uM | ALA2078011 | 5.58 | inhibitor [Ki=2.6uM] | nM | Rattus norvegicus | |
| 5. |  [³H]methotrexate | 138 | Km | = | 4.5 | uM | ALA2077992 | substrate [Km=4.5uM] | nM | Rattus norvegicus | ||
| 6. |  [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Km | = | 33.4 | uM | ALA2076292 | substrate [Km=33.4uM] | nM | Rattus norvegicus | ||
| 7. |  ALA2074644 | Taurolithocholate-3-sulfate | Km | = | 3.06 | uM | ALA2076290 | substrate [Km=3.06uM] | nM | Rattus norvegicus | ||
| 8. | ALA2074644 | Taurolithocholate-3-sulfate | Km | = | 3.06 | uM | ALA2076291 | substrate [Km=3.06uM] | nM | Rattus norvegicus | ||
| 9. |  [³H]taurocholic acid | THCA | Km | = | 15.9 | uM | ALA2076290 | substrate [Km=15.9uM] | nM | Rattus norvegicus | ||
| 10. |  MK 571 sodium salt (L 660711 sodium salt) | Mk-679 | Activity | = | 9.5 | % | ALA2078008 | inhibitor [9.5% of control] | % | Rattus norvegicus | ||
| 11. | [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Activity | = | 78.4 | % | ALA2078000 | inhibitor [78.4% of control] | % | Rattus norvegicus | ||
| 12. | [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Activity | = | 78.4 | % | ALA2077999 | inhibitor [78.4 % of control] | % | Rattus norvegicus | ||
| 13. |  ALA495936 | Leukotriene C4 (LTC4) | Activity | = | 57 | % | ALA2078014 | inhibitor [57 % of control] | % | Rattus norvegicus | ||
| 14. | MK 571 sodium salt (L 660711 sodium salt) | Mk-679 | Activity | = | 4.9 | % | ALA2078007 | inhibitor [4.9% of control] | % | Rattus norvegicus | ||
| 15. |  estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Activity | = | 33.3 | % | ALA2078016 | inhibitor [33.3 % of control] | % | Rattus norvegicus | ||
| 16. |  ALA2074736 | Taurochenodeoxycholate sulfate | Activity | = | 27.8 | % | ALA2078002 | inhibitor [27.8% of control] | % | Rattus norvegicus | ||
| 17. | ALA2074736 | Taurochenodeoxycholate sulfate | Activity | = | 27.8 | % | ALA2077997 | inhibitor [27.8% of control] | % | Rattus norvegicus | ||
| 18. | ALA2074736 | Taurochenodeoxycholate sulfate | Activity | = | 26.2 | % | ALA2077974 | inhibitor [26.2% of control] | % | Rattus norvegicus | ||
| 19. | ALA2074736 | Taurochenodeoxycholate sulfate | Activity | = | 26.2 | % | ALA2078020 | inhibitor [26.2 % of control] | % | Rattus norvegicus | ||
| 20. |  1-Naphthol β-D-glucuronide | alpha-naphthyl beta-D-glucuronide | Activity | = | 23.6 | % | ALA2078012 | inhibitor [23.6 % of control] | % | Rattus norvegicus |
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