# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1651104 | 7 | INH | = | 50 | % | ALA3382980 | % | Homo sapiens | |||
2. | ALA1651100 | 2 | INH | = | 50 | % | ALA3382980 | % | Homo sapiens | |||
3. | Cepharanthine | 12 | INH | = | 20 | % | ALA3382979 | % | Homo sapiens | |||
4. | ALA1651099 | 1 | INH | 0 | ALA3382977 | Not Active | % | Homo sapiens | ||||
5. | ALA1651105 | 9 | INH | 0 | ALA3382977 | Not Active | % | Homo sapiens | ||||
6. | ALA1651104 | 7 | INH | = | 40 | % | ALA3382976 | % | Homo sapiens | |||
7. | ALA1651100 | 2 | INH | = | 40 | % | ALA3382975 | % | Homo sapiens | |||
8. | [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | Km | = | 57.8 | uM | ALA2076521 | substrate [Km=57.8uM] | nM | Homo sapiens | ||
9. | [³H]methotrexate | 138 | Activity | = | 74 | % | ALA2076674 | inhibitor [74 % of control] | % | Homo sapiens | ||
10. | β-Estradiol | Table II | Activity | = | 60.7 | % | ALA2076522 | inhibitor [60.7 % of control] | % | Homo sapiens | ||
11. | ALA1236070 | 16alpha,17beta-Estriol 3-(beta-D-glucuronide) | Activity | = | 58.5 | % | ALA2077025 | inhibitor [58.5 % of control] | % | Homo sapiens | ||
12. | Glycocholic acid | 5b, glyco | Activity | = | 58.4 | % | ALA2077857 | inhibitor [58.4 % of control] | % | Homo sapiens | ||
13. | Estriol 16α-(β-D-glucuronide) | 16alpha,17beta-Estriol 16-(beta-D-glucuronide) | Activity | = | 53 | % | ALA2077026 | inhibitor [53 % of control] | % | Homo sapiens | ||
14. | Cyclosporin A | 1a Cys-A | Activity | = | 49.6 | % | ALA2077022 | inhibitor [49.6 % of control] | % | Homo sapiens | ||
15. | Etoposide | VP-16 | Activity | = | 49.5 | % | ALA2076669 | inhibitor [49.5 % of control] | % | Homo sapiens | ||
16. | ALA2074797 | 16alpha,17beta-Estriol 3-sulfate | Activity | = | 49.4 | % | ALA2077024 | inhibitor [49.4 % of control] | % | Homo sapiens | ||
17. | ALA28079 | M&B-22948 | Activity | = | 48.3 | % | ALA2076523 | inhibitor [48.3 % of control] | % | Homo sapiens | ||
18. | ALA213947 | M2 | Activity | = | 46.4 | % | ALA2077021 | inhibitor [46.4 % of control] | % | Homo sapiens | ||
19. | [³H]taurocholic acid | THCA | Activity | = | 44.5 | % | ALA2076672 | inhibitor [44.5 % of control] | % | Homo sapiens | ||
20. | ALA285913 | Trequinsin | Activity | = | 44.3 | % | ALA2076670 | inhibitor [44.3 % of control] | % | Homo sapiens |