| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Ki | = | 53.1 | uM | ALA2078136 | 4.28 | inhibitor [Ki=53.1 +/- 7.4uM] | nM | Mus musculus | |
| 2. |  Probenecid | probenecid | Ki | = | 293 | uM | ALA2078136 | inhibitor [Ki=293 +/- 115uM] | nM | Mus musculus | ||
| 3. |  3,3',5-Triiodo-L-thyronine | 11 | Ki | = | 24.2 | uM | ALA2078136 | 4.62 | inhibitor [Ki=24.2 +/- 9.7uM] | nM | Mus musculus | |
| 4. |  3,3′,5-Triiodothyroacetic acid | 3 | Ki | = | 2.15 | uM | ALA2078136 | 5.67 | inhibitor [Ki=2.15 +/- 0.50uM] | nM | Mus musculus | |
| 5. |  [³H]taurocholic acid | THCA | Ki | = | 109 | uM | ALA2078136 | inhibitor [Ki=109 +/- 32uM] | nM | Mus musculus | ||
| 6. |  3,3′,5′-Triiodo-L-thyronine | reverse tri-iodothyronine (r-T3) | Ki | = | 0.91 | uM | ALA2078136 | 6.04 | inhibitor [Ki=0.91 +/- 0.21uM] | nM | Mus musculus | |
| 7. |  D-Thyroxine | 12 | Ki | = | 0.27 | uM | ALA2078136 | 6.57 | inhibitor [Ki=0.27 +/- 0.04uM] | nM | Mus musculus | |
| 8. |  17β-Estradiol 17β-D-Glucuronide | estradiol 17b glucuronide | Ki | > | 100 | uM | ALA2078136 | inhibitor [Ki >100uM] | nM | Mus musculus | ||
| 9. | 17β-Estradiol 17β-D-Glucuronide | estradiol 17b glucuronide | Km | = | 23.5 | ALA2076875 | substrate [Km=23.5 +/- 5.2] | Mus musculus | ||||
| 10. | 3,3′,5′-Triiodo-L-thyronine | reverse tri-iodothyronine (r-T3) | Km | = | 0.46 | ALA2076875 | substrate [Km=0.46 +/- 0.08] | Mus musculus | ||||
| 11. |  L-Thyroxine | 181 (Thyroxine) | Km | = | 0.34 | ALA2076875 | substrate [Km=0.34 +/- 0.03] | Mus musculus |
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