# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4460144 | JBP923 | Ratio | = | 7.3 | ALA4375692 | Rattus norvegicus | |||||
2. | ALA4540326 | 12a; J3V | Ratio | = | 6.8 | ALA4375692 | Rattus norvegicus | |||||
3. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Ratio | = | 2.5 | ALA4375692 | Rattus norvegicus | |||||
4. | ALA4540326 | 12a; J3V | Ratio | = | 6.03 | ALA4375691 | Rattus norvegicus | |||||
5. | ALA4460144 | JBP923 | Peff | 0 | ALA4375690 | Permeable | Rattus norvegicus | |||||
6. | ALA4540326 | 12a; J3V | Peff | 0 | ALA4375690 | Permeable | Rattus norvegicus | |||||
7. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Peff | 0 | ALA4375690 | Permeable | Rattus norvegicus | |||||
8. | ALA3707141 | [3H]-GlySar | FC | = | 100 | ALA3538387 | Rattus norvegicus | |||||
9. | ALA3707141 | [3H]-GlySar | FC | = | 136 | ALA3538390 | Rattus norvegicus | |||||
10. | ALA3707141 | [3H]-GlySar | Vmax | = | 88.8 | pmol/OD/min | ALA3540999 | pmol/OD/min | Rattus norvegicus | |||
11. | ALA3707141 | [3H]-GlySar | Km | = | 0.16 | mM | ALA3540999 | nM | Rattus norvegicus | |||
12. | ALA3707141 | [3H]-GlySar | Kd | = | 2.21 | uL/OD/min | ALA3541258 | uL/OD/min | Rattus norvegicus | |||
13. | ALA3707141 | [3H]-GlySar | Vmax/Km | = | 555 | uL/OD/min | ALA3541261 | uL/OD/min | Rattus norvegicus | |||
14. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 100 | % | ALA3541264 | % | Rattus norvegicus | |||
15. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 91.5 | % | ALA3541267 | % | Rattus norvegicus | |||
16. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 113 | % | ALA3541270 | % | Rattus norvegicus | |||
17. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 0.6 | % | ALA3541273 | % | Rattus norvegicus | |||
18. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 23.1 | % | ALA3541276 | % | Rattus norvegicus | |||
19. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 23.4 | % | ALA3530856 | % | Rattus norvegicus | |||
20. | ALA3707141 | [3H]-GlySar | Drug uptake | = | 93.7 | % | ALA3530859 | % | Rattus norvegicus |