# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [³H]taurocholic acid | THCA | Km | = | 72 | uM | ALA2212536 | nM | Rattus norvegicus | |||
2. | Dehydroepiandrosterone sulfate | Dehydroepiandrosterone sulfate (DHEAS) | Activity | 0 | ALA2076810 | is not a substrate [-] | Rattus norvegicus | |||||
3. | Digoxin | Digoxin | Activity | 0 | ALA2076810 | is not a substrate [-] | Rattus norvegicus | |||||
4. | Dinoprost | 9 | Activity | 0 | ALA2076810 | is not a substrate [-] | Rattus norvegicus | |||||
5. | Dinoprost | 9 | IC50 | = | 0.287 | uM | ALA2075311 | 6.54 | inhibitor [IC50=0.287uM] | nM | Rattus norvegicus | |
6. | Prostaglandin E1 | PGE1 | IC50 | = | 0.036 | uM | ALA2075311 | 7.45 | inhibitor [IC50=0.0358uM] | nM | Rattus norvegicus | |
7. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 3.2 | uM | ALA2076810 | substrate [Km=3.2uM] | nM | Rattus norvegicus | ||
8. | [³H]taurocholic acid | THCA | Km | = | 17.6 | uM | ALA2076810 | substrate [Km=17.6uM] | nM | Rattus norvegicus | ||
9. | Iloprost | Iloprost | Activity | 0 | ALA2076810 | substrate [+] | Rattus norvegicus | |||||
10. | Prostaglandin E1 | PGE1 | Activity | 0 | ALA2076810 | substrate [+] | Rattus norvegicus | |||||
11. | Prostaglandin E₂ | PGE2 | Activity | 0 | ALA2076810 | substrate [+] | Rattus norvegicus | |||||
12. | Thromboxane B2 | SID26754848 | Activity | 0 | ALA2076810 | substrate [+] | Rattus norvegicus | |||||
13. | [³H]PGD₂ | SID26754808 | Km | = | 0.036 | uM | ALA2076810 | substrate [Km=0.0355uM] | nM | Rattus norvegicus |