Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA2387397	45	IC50	=	0.3	nM	ALA2388853	9.52		nM	Mus musculus
2.	ALA2385105	20	IC50	=	0.5	nM	ALA2388853	9.30		nM	Mus musculus
3.	ALA2387399	47	IC50	=	0.9	nM	ALA2388853	9.05		nM	Mus musculus
4.	(3R,5R)-3-butyl-3-ethyl-7,8-dimethoxy-5-phenyl-4,5-dihydro-2H-benzo[f][1,4]thiazepine 1,1-dioxide	2	IC50	=	3	nM	ALA2388853	8.52		nM	Mus musculus
5.	ALA2387419	44	IC50		0		ALA2388853		Not Determined		Mus musculus
6.	ALA2387402	50	IC50		0		ALA2388853		Not Determined		Mus musculus
7.	Linerixibat	56, GSK2330672	IC50	=	2.1	nM	ALA2388853	8.68		nM	Mus musculus
8.	ALA2074988	2164U90	Ki	=	0.068	uM	ALA2075491	7.17	inhibitor [Ki=0.068uM]	nM	Mus musculus
9.	[³H]taurocholic acid	THCA	Km	=	27	uM	ALA2075485		substrate [Km=27uM]	nM	Mus musculus
10.	Lithocholic acid	LCA	Activity		0		ALA2075487		inhibitor [+]		Mus musculus
11.	Glycocholic acid	5b, glyco	Activity		0		ALA2075488		inhibitor [+]		Mus musculus
12.	Deoxycholic acid	7, DCA	Activity		0		ALA2076337		inhibitor [+]		Mus musculus
13.	Deoxycholic acid	7, DCA	Activity		0		ALA2076337		inhibitor [+]		Mus musculus
14.	Chenodeoxycholic acid	1	Activity		0		ALA2075489		inhibitor [+]		Mus musculus
15.	[³H]taurocholic acid	THCA	Activity		0		ALA2075490		inhibitor [+]		Mus musculus
16.	[³H]taurocholic acid	THCA	Km	=	13	uM	ALA2075486		substrate [Km=13uM]	nM	Mus musculus
17.	ALA4202981	12	pIC50	<	4.6		ALA4200891			nM	Mus musculus
18.	ALA4217797	64	pIC50	<	4.6		ALA4200891			nM	Mus musculus
19.	ALA4205214	25	pIC50	<	4.6		ALA4200891			nM	Mus musculus