# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3186763 | SID144087340 | INH | = | 10.78 | % | ALA3383685 | % | Rattus norvegicus | |||
2. | ALA4283703 | (+/-)-1 | Ki | = | 1.1 | nM | ALA4256526 | 8.96 | nM | Rattus norvegicus | ||
3. | ALA4290888 | (2aR,4aS,9aS)-1 | Ki | = | 0.87 | nM | ALA4256526 | 9.06 | nM | Rattus norvegicus | ||
4. | ALA1086654 | 4 | Ki | = | 29 | nM | ALA4256526 | 7.54 | nM | Rattus norvegicus | ||
5. | ALA1199383 | 3 | Ki | = | 11 | nM | ALA4256526 | 7.96 | nM | Rattus norvegicus | ||
6. | (±)-Epibatidine | 9 | Ki | = | 0.041 | nM | ALA4256526 | 10.39 | nM | Rattus norvegicus | ||
7. | (±)-Epibatidine | 9 | Ratio Ki | = | 25 | ALA4256527 | Rattus norvegicus | |||||
8. | ALA1181055 | 6 | Kd | = | 2.2 | nM | ALA4178950 | 8.66 | nM | Rattus norvegicus | ||
9. | Anabasine | table I | Inhibition | = | 91 | % | ALA633999 | % | Rattus norvegicus | |||
10. | Anabasine | table I | Kd | = | 0.001 | M | ALA632853 | nM | Rattus norvegicus | |||
11. | Anabasine | table I | Kd | = | 0 | M | ALA634000 | 5.58 | nM | Rattus norvegicus | ||
12. | ALA15722 | beta-picoline | Inhibition | = | 121 | % | ALA633999 | % | Rattus norvegicus | |||
13. | ALA15722 | beta-picoline | Kd | = | 0.002 | M | ALA634000 | nM | Rattus norvegicus | |||
14. | mecamylamine | 2a | Mean enhancement of binding | = | 16.4 | ALA638619 | Rattus norvegicus | |||||
15. | mecamylamine | 2a | Enhancement | = | 20 | % | ALA874428 | % | Rattus norvegicus | |||
16. | 4-Hydroxy-1-methylpiperidine | table I | Mean enhancement of binding | = | 13 | ALA639522 | Rattus norvegicus | |||||
17. | 4-Hydroxy-1-methylpiperidine | table I | Inhibition | = | 88 | % | ALA633999 | % | Rattus norvegicus | |||
18. | 4-Hydroxy-1-methylpiperidine | table I | Enhancement | = | 20 | % | ALA874428 | % | Rattus norvegicus | |||
19. | 4-Hydroxy-1-methylpiperidine | table I | Kd | = | 0.003 | M | ALA632853 | nM | Rattus norvegicus | |||
20. | 4-Hydroxy-1-methylpiperidine | table I | Kd | < | 0 | M | ALA634001 | nM | Rattus norvegicus |