# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3250939 | 1 | INH | 0 | ALA3257671 | Not Active | % | Rattus norvegicus | ||||
2. | ALA3250942 | 5 | INH | 0 | ALA3257670 | Active | % | Rattus norvegicus | ||||
3. | ALA404594 | 16 | pA2 | = | 8.6 | ALA3256389 | 8.60 | nM | Rattus norvegicus | |||
4. | ALA3249921 | [Sar1,Sar7,DL-aIle8]AII | pA2 | = | 8.4 | ALA3256389 | 8.40 | nM | Rattus norvegicus | |||
5. | ALA3249557 | [Sar1,Sar7,Thr(Me)8]AII | pA2 | = | 7.4 | ALA3256389 | 7.40 | nM | Rattus norvegicus | |||
6. | ALA3249556 | [Sar1,Sar7,Met8]AII | pA2 | = | 7.7 | ALA3256389 | 7.70 | nM | Rattus norvegicus | |||
7. | ALA3249555 | [Sar1,Sar7,Ala8]AII | pA2 | = | 7 | ALA3256389 | 7.00 | nM | Rattus norvegicus | |||
8. | ALA3244481 | [Sar1,Sar7,Leu8]AII | pA2 | = | 7.4 | ALA3256389 | 7.40 | nM | Rattus norvegicus | |||
9. | ALA3249554 | [Sar1,Sar7,Ile8]AII | pA2 | = | 8.1 | ALA3256389 | 8.10 | nM | Rattus norvegicus | |||
10. | ALA404594 | 16 | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
11. | ALA3249921 | [Sar1,Sar7,DL-aIle8]AII | Intrinsic activity | = | 0.7 | % | ALA3256388 | % | Rattus norvegicus | |||
12. | ALA3249557 | [Sar1,Sar7,Thr(Me)8]AII | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
13. | ALA3249556 | [Sar1,Sar7,Met8]AII | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
14. | ALA3249555 | [Sar1,Sar7,Ala8]AII | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
15. | ALA3244481 | [Sar1,Sar7,Leu8]AII | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
16. | ALA3249554 | [Sar1,Sar7,Ile8]AII | Intrinsic activity | < | 0.1 | % | ALA3256388 | % | Rattus norvegicus | |||
17. | ALA3249553 | [Sar1,Sar7]AII | Intrinsic activity | = | 22 | % | ALA3256388 | % | Rattus norvegicus | |||
18. | ALA3247675 | Oct-LAT, Octanoyl[8-leucyl]angiotensin II | Activity | = | 0.21 | % | ALA3258706 | % | Rattus norvegicus | |||
19. | ALA3247163 | 11 | Activity | = | 0.025 | % | ALA3258706 | % | Rattus norvegicus | |||
20. | ALA3247675 | Oct-LAT, Octanoyl[8-leucyl]angiotensin II | t1/2 | = | 6.6 | min | ALA3255082 | hr | Rattus norvegicus |