# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5268786 | 264; RPR-200765A | IC50 | = | 50 | nM | ALA5247061 | 7.30 | nM | Homo sapiens | ||
2. | ALA5290093 | 263; RPR-201227A | IC50 | = | 44 | nM | ALA5247061 | 7.36 | nM | Homo sapiens | ||
3. | SB 203580 (DMSO solution) | 9 | IC50 | = | 56 | nM | ALA5247061 | 7.25 | nM | Homo sapiens | ||
4. | ALA5275239 | 47 | INH | = | 37 | % | ALA5236715 | % | Homo sapiens | |||
5. | ALA5275239 | 47 | INH | = | 99 | % | ALA5236714 | % | Homo sapiens | |||
6. | ALA5193786 | 34b | IC50 | > | 30 | uM | ALA5166095 | nM | Homo sapiens | |||
7. | ALA5189796 | 6b; EB1 | INH | 0 | ALA5164573 | NA | % | Homo sapiens | ||||
8. | SB 203580 (DMSO solution) | 9 | IC50 | = | 0.3 | uM | ALA5131859 | 6.52 | nM | Homo sapiens | ||
9. | Nilotinib (AMN-107) | 38 | INH | 0 | ALA5120291 | Active | % | Homo sapiens | ||||
10. | Nilotinib (AMN-107) | 38 | INH | 0 | ALA5120290 | Active | % | Homo sapiens | ||||
11. | Nilotinib (AMN-107) | 38 | Activity | 0 | ALA5120262 | Active | Homo sapiens | |||||
12. | ALA4550547 | SW083604 | deltaTm | = | 0.3 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
13. | ALA4537058 | SW034538 | deltaTm | = | 2.8 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
14. | ALA3715362 | 39 | deltaTm | = | 2 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
15. | ALA4586284 | SW172006 | deltaTm | = | 2 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
16. | ALA4553877 | SW163112 | deltaTm | = | 1.5 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
17. | ALA4554066 | SW106178 | deltaTm | = | 1.3 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
18. | ALA1700355 | SID56432189 | deltaTm | = | 2 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
19. | ALA4567815 | SW166693 | deltaTm | = | 0 | degrees C | ALA4479298 | degrees C | Homo sapiens | |||
20. | ALA1448756 | SID4263243 | deltaTm | = | 2.2 | degrees C | ALA4479298 | degrees C | Homo sapiens |