# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2113483 | 5 | EC50 | = | 367 | nM | ALA649127 | 6.43 | nM | Rattus norvegicus | ||
2. | ALA2113483 | 5 | Ki | = | 9.1 | nM | ALA649868 | 8.04 | nM | Rattus norvegicus | ||
3. | ALA2113449 | 4 | EC50 | = | 440 | nM | ALA649127 | 6.36 | nM | Rattus norvegicus | ||
4. | ALA2113449 | 4 | Ki | = | 57.8 | nM | ALA649868 | 7.24 | nM | Rattus norvegicus | ||
5. | ALA2113399 | 15 | EC50 | = | 456 | nM | ALA649127 | 6.34 | nM | Rattus norvegicus | ||
6. | ALA2113399 | 15 | Ki | = | 1.7 | nM | ALA649868 | 8.77 | nM | Rattus norvegicus | ||
7. | RX821002 | 31 | Antagonist potency | = | 2 | ALA650234 | Rattus norvegicus | |||||
8. | RX821002 | 31 | Antagonist potency | = | 2.9 | ALA650233 | Rattus norvegicus | |||||
9. | RX821002 | 31 | Antagonist potency | = | 4.7 | ALA650235 | Rattus norvegicus | |||||
10. | RX821002 | 31 | Antagonist potency | = | 1 | ALA650236 | Rattus norvegicus | |||||
11. | RX821002 | 31 | Antagonist potency | = | 15.5 | ALA650232 | Rattus norvegicus | |||||
12. | ALA2113403 | 18 | EC50 | = | 564 | nM | ALA649127 | 6.25 | nM | Rattus norvegicus | ||
13. | ALA2113403 | 18 | Ki | = | 38.3 | nM | ALA649868 | 7.42 | nM | Rattus norvegicus | ||
14. | RX821002 | 31 | Antagonist potency | = | 1836 | ALA650234 | Rattus norvegicus | |||||
15. | RX821002 | 31 | Antagonist potency | = | 1620 | ALA650233 | Rattus norvegicus | |||||
16. | RX821002 | 31 | Antagonist potency | = | 972 | ALA650235 | Rattus norvegicus | |||||
17. | RX821002 | 31 | Antagonist potency | = | 544 | ALA650236 | Rattus norvegicus | |||||
18. | RX821002 | 31 | Antagonist potency | = | 0.037 | ALA650232 | Rattus norvegicus | |||||
19. | [³H]CCPA | CCPA | EC50 | > | 10 | uM | ALA649127 | nM | Rattus norvegicus | |||
20. | [³H]CCPA | CCPA | Ki | = | 650 | nM | ALA649868 | 6.19 | nM | Rattus norvegicus |