# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA479683 | 1 | INH | = | 17.4 | % | ALA3129970 | % | Homo sapiens | |||
2. | PF 04418948 | 15, PF-04418948 | % inhibition | 1 | % | ALA4887027 | Not Active | % | Homo sapiens | |||
3. | ALA4536197 | EUB0000326 | % inhibition | 2 | % | ALA4886759 | Not Active | % | Homo sapiens | |||
4. | A 485 | A-485 | % inhibition | 4 | % | ALA4886554 | Not Active | % | Homo sapiens | |||
5. | ALA3480577 | DDD01251909 | pKi | 6 | ALA4880069 | nM | Homo sapiens | |||||
6. | ALA3480577 | DDD01251909 | Ki | 1004 | nM | ALA4880069 | nM | Homo sapiens | ||||
7. | ALA3480577 | DDD01251909 | % Inhibition | 0 | % | ALA4880069 | Not Active | % | Homo sapiens | |||
8. | PF-04457845 | 23, PF-04457845 | % inhibition | -3 | % | ALA4883114 | Not Active | % | Homo sapiens | |||
9. | ALA3298233 | 7m | Activity | 0 | ALA3367434 | Not Active | Homo sapiens | |||||
10. | ALA2206397 | 6d, Ro-4992479 | INH | = | 2 | % | ALA2216407 | % | Homo sapiens | |||
11. | L-Glutamic acid polymer | Glutamic acid | IC50 | = | 70 | nM | ALA2208698 | 7.16 | nM | Homo sapiens | ||
12. | ALA1205743 | Table 32, R1C1 | IC50 | = | 2.3 | uM | ALA2208698 | 5.64 | nM | Homo sapiens | ||
13. | ALA1207193 | Table 32, R2C1 | IC50 | = | 1.6 | uM | ALA2208698 | 5.80 | nM | Homo sapiens | ||
14. | ALA1205735 | Table 32, R3C1 | IC50 | = | 10 | uM | ALA2208698 | 5.00 | nM | Homo sapiens | ||
15. | ALA145806 | 26 | IC50 | = | 0.47 | uM | ALA2208698 | 6.33 | nM | Homo sapiens | ||
16. | ALA4865171 | (2S,6R)-3f | INH | = | 7 | % | ALA4818782 | % | Homo sapiens | |||
17. | ALA4866255 | (2S,6R)-3g | INH | = | 14 | % | ALA4818782 | % | Homo sapiens | |||
18. | ALA4857800 | (2R,6S)-3g | INH | = | 43 | % | ALA4818782 | % | Homo sapiens | |||
19. | ALA4865545 | (2S,6R)-3d | INH | = | 37 | % | ALA4818782 | % | Homo sapiens | |||
20. | ALA4853884 | (2R,6S)-3d | INH | = | 31 | % | ALA4818782 | % | Homo sapiens |