# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY-091 | EUB0001564 | % inhibition | 7.13 | % | ALA4887805 | Not Active | % | Homo sapiens | |||
2. | ALA2180408 | Figure 27, R1C1 | % inhibition | 1 | % | ALA4886202 | Not Active | % | Homo sapiens | |||
3. | ALA4580220 | EUB0000311 | % residual kinase activity | 92 | % | ALA4884248 | Not Active | % | Homo sapiens | |||
4. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 85 | % | ALA4883852 | Not Active | % | Homo sapiens | |||
5. | TC-S 7001 | SID103905649 | % inhibition | 40 | % | ALA4881499 | Not Active | % | Homo sapiens | |||
6. | BAY-885 | BAY-885; 41 | % residual kinase activity | 99 | % | ALA4880984 | Not Active | % | Homo sapiens | |||
7. | 2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | 9 | % | ALA4880585 | Not Active | % | Homo sapiens | |||
8. | ALA280074 | Olomoucine | IC50 | = | 5 | ug ml-1 | ALA5262854 | ug.mL-1 | Homo sapiens | |||
9. | ALA5287185 | 80 | IC50 | = | 4 | ug ml-1 | ALA5262854 | ug.mL-1 | Homo sapiens | |||
10. | ALA5288780 | 79 | IC50 | = | 4 | ug ml-1 | ALA5262854 | ug.mL-1 | Homo sapiens | |||
11. | ALA5278558 | 76 | IC50 | = | 4 | ug ml-1 | ALA5262854 | ug.mL-1 | Homo sapiens | |||
12. | ALA5285888 | 74 | IC50 | = | 4 | ug ml-1 | ALA5262854 | ug.mL-1 | Homo sapiens | |||
13. | ALA5285374 | 31 | IC50 | = | 3.8 | uM | ALA5262854 | 5.42 | nM | Homo sapiens | ||
14. | ALA5279668 | 30 | IC50 | = | 3.8 | uM | ALA5262854 | 5.42 | nM | Homo sapiens | ||
15. | ALA5281814 | 29 | IC50 | = | 3.8 | uM | ALA5262854 | 5.42 | nM | Homo sapiens | ||
16. | ALA5279829 | 28 | IC50 | = | 5 | uM | ALA5262854 | 5.30 | nM | Homo sapiens | ||
17. | ALA5285775 | 27 | IC50 | = | 3.8 | uM | ALA5262854 | 5.42 | nM | Homo sapiens | ||
18. | PF-06873600 | PF-06873600 | IC50 | = | 0.02 | uM | ALA5259479 | 7.70 | nM | Homo sapiens | ||
19. | ALA5288714 | 23 | IC50 | = | 1.6 | uM | ALA5259479 | 5.80 | nM | Homo sapiens | ||
20. | ALA5275414 | KII-22 | IC50 | = | 0.92 | uM | ALA5259479 | 6.04 | nM | Homo sapiens |