# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4802042 | EUB0001568 | % inhibition | 0 | % | ALA4888341 | Not Active | % | Homo sapiens | |||
2. | Borussertib | EUB0000645a | % Inhibition | 3 | % | ALA4888168 | Not Active | % | Homo sapiens | |||
3. | BAY-091 | EUB0001564 | % inhibition | 8.82 | % | ALA4888124 | Not Active | % | Homo sapiens | |||
4. | BI 605906 | BI605906 | % Ctrl | 94 | % | ALA4887374 | Not Active | % | Homo sapiens | |||
5. | BI 605906 | BI605906 | % Ctrl | 92 | % | ALA4887374 | Not Active | % | Homo sapiens | |||
6. | ALA2180408 | Figure 27, R1C1 | % inhibition | 5 | % | ALA4886200 | Not Active | % | Homo sapiens | |||
7. | ALA4475494 | 19 | % Inhibition | 2.5 | % | ALA4885924 | Not Active | % | Homo sapiens | |||
8. | ALA4580220 | EUB0000311 | % residual kinase activity | 98 | % | ALA4884246 | Not Active | % | Homo sapiens | |||
9. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 83 | % | ALA4883849 | Not Active | % | Homo sapiens | |||
10. | CLK-IN-T3 | EUB0000321 | % inhibition | 7.946 | % | ALA4883226 | Not Active | % | Homo sapiens | |||
11. | CLK-IN-T3 | EUB0000321 | % inhibition | 7.102 | % | ALA4883226 | Not Active | % | Homo sapiens | |||
12. | MLI-2 | 1; MLi-2 | % Inhibition | 1.293 | % | ALA4882679 | Not Active | % | Homo sapiens | |||
13. | 4-[[[5-(2-ethoxycarbonyl-1H-indol-5-yl)-1-methylpyrazole-3-carbonyl]amino]methyl]benzoic acid | 15 | % Ctrl | 88 | % | ALA4882428 | Not Active | % | Homo sapiens | |||
14. | ALA3417525 | 69, BI665915 | % Ctrl | 99 | % | ALA4881908 | Not Active | % | Homo sapiens | |||
15. | TC-S 7001 | SID103905649 | % inhibition | -22 | % | ALA4881497 | Not Active | % | Homo sapiens | |||
16. | BAY 293 | EUB0000320 | % residual kinase activity | 87 | % | ALA4881464 | Not Active | % | Homo sapiens | |||
17. | BAY-885 | BAY-885; 41 | % residual kinase activity | 101 | % | ALA4880982 | Not Active | % | Homo sapiens | |||
18. | 2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | 16 | % | ALA4880584 | Not Active | % | Homo sapiens | |||
19. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 2.52 | nM | ALA3620022 | 8.60 | nM | Homo sapiens | ||
20. | ALA3616990 | Page 600, C2, R16 | INH | 0 | ALA3619887 | Not Active | % | Homo sapiens |