# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | A-1155463 | 17, A-1155463 | % of inhibition | = | 98.9 | % | ALA5213783 | % | Homo sapiens | |||
2. | A-1155463 | 17, A-1155463 | % of inhibition | = | 98.9 | % | ALA5213782 | % | Homo sapiens | |||
3. | ALA5177923 | Leu15-gastrin-17 | EC50 | > | 100 | nM | ALA5146165 | nM | Homo sapiens | |||
4. | ALA5205878 | xGLP-1 | EC50 | 0 | ALA5146165 | ND | Homo sapiens | |||||
5. | ALA410972 | 1 | EC50 | 0 | ALA5146165 | ND | Homo sapiens | |||||
6. | ALA5182775 | 2d | EC50 | = | 1.03 | nM | ALA5146165 | 8.99 | nM | Homo sapiens | ||
7. | ALA5182331 | 2c | EC50 | = | 0.83 | nM | ALA5146165 | 9.08 | nM | Homo sapiens | ||
8. | ALA5182323 | 2b | EC50 | = | 1.19 | nM | ALA5146165 | 8.92 | nM | Homo sapiens | ||
9. | ALA5181266 | 2a | EC50 | = | 1.25 | nM | ALA5146165 | 8.90 | nM | Homo sapiens | ||
10. | ALA5185239 | 1b | EC50 | = | 0.95 | nM | ALA5146165 | 9.02 | nM | Homo sapiens | ||
11. | ALA5182173 | 1a | EC50 | = | 1.14 | nM | ALA5146165 | 8.94 | nM | Homo sapiens | ||
12. | ALA4440419 | 9; NN9056 | EC50 | = | 0.21 | nM | ALA5146165 | 9.68 | nM | Homo sapiens | ||
13. | ML417 | 20; ML417 | INH | = | 63 | % | ALA4406557 | % | Homo sapiens | |||
14. | ALA4579120 | 40; E40 | INH | = | 61.4 | % | ALA4396166 | % | Homo sapiens | |||
15. | ALA4540275 | 6 | IC50 | < | 50 | nM | ALA4394889 | nM | Homo sapiens | |||
16. | RK-287107 | 1; RK-287107 | INH | > | 20 | % | ALA4388183 | % | Homo sapiens | |||
17. | ALA4518377 | Page no 1411, R62C2, cpd 3-(31-Ser) | pEC50 | 0 | ALA4370032 | Not Active | Homo sapiens | |||||
18. | ALA4473611 | Page no 1411, R62C2, cpd 3-(31-Ala) | pEC50 | 0 | ALA4370032 | Not Active | Homo sapiens | |||||
19. | ALA4454469 | Page no 1411, R62C2, cpd 3-(31-Lys) | pEC50 | 0 | ALA4370032 | Not Active | Homo sapiens | |||||
20. | ALA4564249 | Page no 1411, R63C2, cpd 3-(31-Glu) | pEC50 | 0 | ALA4370032 | Not Active | Homo sapiens |