# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4065991 | 4d | Ki | > | 100 | uM | ALA4415161 | nM | Homo sapiens | |||
2. | 5-(N,N-hexamethylene)-amiloride | 5m | IC50 | = | 0.27 | uM | ALA3821345 | 6.57 | nM | Homo sapiens | ||
3. | ALA3819313 | 12h | IC50 | = | 0.12 | uM | ALA3821345 | 6.92 | nM | Homo sapiens | ||
4. | ALA3818888 | 12i | IC50 | = | 0.25 | uM | ALA3821345 | 6.60 | nM | Homo sapiens | ||
5. | ALA3818205 | 12k | IC50 | = | 0.07 | uM | ALA3821345 | 7.16 | nM | Homo sapiens | ||
6. | ALA3818905 | 12l | IC50 | = | 0.05 | uM | ALA3821345 | 7.30 | nM | Homo sapiens | ||
7. | 5-(N,N-hexamethylene)-amiloride | 5m | Time | = | 1.4 | min | ALA3821346 | hr | Homo sapiens | |||
8. | ALA3819313 | 12h | Time | = | 2 | min | ALA3821346 | hr | Homo sapiens | |||
9. | ALA3818888 | 12i | Time | = | 0.8 | min | ALA3821346 | hr | Homo sapiens | |||
10. | ALA3818205 | 12k | Time | = | 1.2 | min | ALA3821346 | hr | Homo sapiens | |||
11. | ALA3818905 | 12l | Time | = | 1.3 | min | ALA3821346 | hr | Homo sapiens | |||
12. | 5-(N,N-hexamethylene)-amiloride | 5m | FC | = | 1.9 | ALA3821475 | Homo sapiens | |||||
13. | ALA3819313 | 12h | FC | = | 1.3 | ALA3821475 | Homo sapiens | |||||
14. | ALA3818888 | 12i | FC | = | 3.4 | ALA3821475 | Homo sapiens | |||||
15. | ALA3818205 | 12k | FC | = | 2.3 | ALA3821475 | Homo sapiens | |||||
16. | ALA3818905 | 12l | FC | = | 2.1 | ALA3821475 | Homo sapiens | |||||
17. | ALA1962823 | 7 | Activity | = | 101 | % | ALA3821343 | % | Homo sapiens | |||
18. | ALA1962615 | 8 | Activity | = | 21 | % | ALA3821343 | % | Homo sapiens | |||
19. | ALA1962848 | 9 | Activity | = | 46 | % | ALA3821343 | % | Homo sapiens | |||
20. | ALA1962616 | 3097 | Activity | = | 73 | % | ALA3821343 | % | Homo sapiens |