# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2431051 | 19 | INH | 0 | ALA2432528 | Not Active | % | Homo sapiens | ||||
2. | ALA15245 | yohimbine | IC50 | = | 5.8 | 10'-8M | ALA2395710 | 7.24 | nM | Homo sapiens | ||
3. | ALA15245 | yohimbine | Ki | = | 2.5 | 10'-8M | ALA2395710 | 7.60 | nM | Homo sapiens | ||
4. | E1R | E1R, 4R,5S-2a | INH | = | -2 | % | ALA2393966 | % | Homo sapiens | |||
5. | ALA15245 | yohimbine | IC50 | = | 36 | nM | ALA2395776 | 7.44 | nM | Homo sapiens | ||
6. | ALA2392692 | 27, GSK2188931B | INH | < | 50 | % | ALA2395866 | % | Homo sapiens | |||
7. | ALA272899 | 1 | Ki | = | 205 | nM | ALA3056598 | 6.69 | nM | Homo sapiens | ||
8. | ALA111612 | 10a | % inhibition | 18 | % | ALA4880241 | Not Active | % | Homo sapiens | |||
9. | ABT-100 | EUB0000289 | % inhibition | < | 10 | % | ALA4880162 | Not Active | % | Homo sapiens | ||
10. | ALA3697701 | BDBM161012 | % inhibition | -1 | % | ALA4880082 | Not Active | % | Homo sapiens | |||
11. | ABT 724 | 3a | % inhibition | 21 | % | ALA4880324 | Not Active | % | Homo sapiens | |||
12. | ALA3408298 | 33, LNP906 | Ki | > | 2240 | nM | ALA3411419 | nM | Homo sapiens | |||
13. | ALA2058635 | 11 | Ki | > | 2500 | nM | ALA3411419 | nM | Homo sapiens | |||
14. | ALA2058631 | 4, LNP 630 | Ki | > | 1949 | nM | ALA3411419 | nM | Homo sapiens | |||
15. | ALA288139 | cis-/trans-1e | Ki | > | 10000 | nM | ALA3411419 | nM | Homo sapiens | |||
16. | ALA3408297 | S 23515 | Ki | > | 10000 | nM | ALA3411419 | nM | Homo sapiens | |||
17. | ALA268734 | B13 | Ki | > | 10000 | nM | ALA3411419 | nM | Homo sapiens | |||
18. | moxonidine | 5 | Ki | = | 75 | nM | ALA3411419 | 7.12 | nM | Homo sapiens | ||
19. | ALA289480 | rilmenidine | Ki | = | 180 | nM | ALA3411419 | 6.75 | nM | Homo sapiens | ||
20. | clonidine | clonidine | Ki | = | 3.8 | nM | ALA3411419 | 8.42 | nM | Homo sapiens |