| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358630 | Not Active | Homo sapiens | |||||
| 2. |  ALA3261926 | 10 | INH | = | 69 | % | ALA3268222 | % | Homo sapiens | |||
| 3. | ALA3261926 | 10 | IC50 | = | 2 | uM | ALA3268220 | 5.70 | nM | Homo sapiens | ||
| 4. |  (S)-ARN2508 | (+)-10r | Activity | = | 1.2 | % | ALA3779487 | % | Homo sapiens | |||
| 5. |  5-(2-Carboxyethyl)-6-[3-[2-ethyl-4-(4-fluorophenyl)-5-hydroxyphenoxy]propoxy]-9-oxoxanthene-2-carboxylic acid | 1 | IC50 | = | 1.2 | nM | ALA699620 | 8.92 | nM | Homo sapiens | ||
| 6. | 5-(2-Carboxyethyl)-6-[3-[2-ethyl-4-(4-fluorophenyl)-5-hydroxyphenoxy]propoxy]-9-oxoxanthene-2-carboxylic acid | 1 | Ki | = | 0.04 | nM | ALA704379 | 10.40 | nM | Homo sapiens | ||
| 7. | 5-(2-Carboxyethyl)-6-[3-[2-ethyl-4-(4-fluorophenyl)-5-hydroxyphenoxy]propoxy]-9-oxoxanthene-2-carboxylic acid | 1 | Ki | = | 0.47 | nM | ALA709860 | 9.33 | nM | Homo sapiens | ||
| 8. |  ALA341757 | 43c | IC50 | = | 7.8 | nM | ALA699620 | 8.11 | nM | Homo sapiens | ||
| 9. | ALA341757 | 43c | Ki | = | 8.4 | nM | ALA704379 | 8.08 | nM | Homo sapiens | ||
| 10. | ALA341757 | 43c | Ki | = | 210 | nM | ALA709860 | 6.68 | nM | Homo sapiens | ||
| 11. |  ALA167972 | 15e | Ki | = | 55 | nM | ALA704379 | 7.26 | nM | Homo sapiens | ||
| 12. | ALA167972 | 15e | Ki | = | 2.9 | nM | ALA709860 | 8.54 | nM | Homo sapiens | ||
| 13. |  ALA88337 | 48 LY-282210 | IC50 | = | 47 | nM | ALA699620 | 7.33 | nM | Homo sapiens | ||
| 14. | ALA88337 | 48 LY-282210 | Ki | = | 1.2 | nM | ALA704379 | 8.92 | nM | Homo sapiens | ||
| 15. | ALA88337 | 48 LY-282210 | Ki | = | 4 | nM | ALA709860 | 8.40 | nM | Homo sapiens | ||
| 16. |  ALA139254 | 56c | IC50 | = | 7.4 | nM | ALA699620 | 8.13 | nM | Homo sapiens | ||
| 17. | ALA139254 | 56c | Ki | = | 11 | nM | ALA704379 | 7.96 | nM | Homo sapiens | ||
| 18. | ALA139254 | 56c | Ki | = | 350 | nM | ALA709860 | 6.46 | nM | Homo sapiens | ||
| 19. |  ALA138954 | 52b | IC50 | = | 2.8 | nM | ALA699620 | 8.55 | nM | Homo sapiens | ||
| 20. | ALA138954 | 52b | Ki | = | 11 | nM | ALA704379 | 7.96 | nM | Homo sapiens |
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