# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5282574 | 36 | Ki | = | 21 | nM | ALA5223230 | 7.68 | nM | Homo sapiens | ||
2. | ALA5288434 | 35 | Ki | = | 99 | nM | ALA5223230 | 7.00 | nM | Homo sapiens | ||
3. | ALA5288617 | 34; BMS-205749 | Ki | = | 5.1 | nM | ALA5223230 | 8.29 | nM | Homo sapiens | ||
4. | ALA2046866 | 33; BMS-193885 | Ki | = | 3.3 | nM | ALA5223230 | 8.48 | nM | Homo sapiens | ||
5. | ALA3787712 | 17 | Kb | = | 25.3 | nM | ALA4478053 | nM | Homo sapiens | |||
6. | ALA4456247 | (R,R)-1 | Kb | = | 9.5 | nM | ALA4478053 | nM | Homo sapiens | |||
7. | ALA4533775 | 22 | Ki | = | 1600 | nM | ALA4478049 | 5.80 | nM | Homo sapiens | ||
8. | ALA4581302 | 21 | Ki | > | 10000 | nM | ALA4478049 | nM | Homo sapiens | |||
9. | ALA4581256 | 20 | Ki | = | 1400 | nM | ALA4478049 | 5.85 | nM | Homo sapiens | ||
10. | ALA4576579 | 19 | Ki | > | 3000 | nM | ALA4478049 | nM | Homo sapiens | |||
11. | ALA3787713 | 18 | Ki | = | 360 | nM | ALA4478049 | 6.44 | nM | Homo sapiens | ||
12. | ALA3787712 | 17 | Ki | = | 410 | nM | ALA4478049 | 6.39 | nM | Homo sapiens | ||
13. | ALA3787766 | 16 | Ki | = | 720 | nM | ALA4478049 | 6.14 | nM | Homo sapiens | ||
14. | ALA4549208 | (2S,7S)-10 | Ki | = | 290 | nM | ALA4478049 | 6.54 | nM | Homo sapiens | ||
15. | ALA4522438 | (2R,7R)-10 | Ki | = | 400 | nM | ALA4478049 | 6.40 | nM | Homo sapiens | ||
16. | ALA4475071 | (S,S)-1 | Ki | = | 930 | nM | ALA4478049 | 6.03 | nM | Homo sapiens | ||
17. | ALA4456247 | (R,R)-1 | Ki | = | 440 | nM | ALA4478049 | 6.36 | nM | Homo sapiens | ||
18. | ALA4436741 | (S,S)-12 | pIC50 | = | 6.63 | ALA4426106 | 6.63 | nM | Homo sapiens | |||
19. | ALA4445077 | (S,S)-9 | pIC50 | = | 6.31 | ALA4426106 | 6.31 | nM | Homo sapiens | |||
20. | ALA4456247 | (R,R)-1 | pIC50 | = | 6.44 | ALA4426106 | 6.44 | nM | Homo sapiens |