| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2204341 | 65 | INH | < | 50 | % | ALA2317819 | % | Homo sapiens | |||
| 2. |  ALA2311601 | 61 | INH | < | 50 | % | ALA2317819 | % | Homo sapiens | |||
| 3. |  ALA2311600 | 62 | INH | < | 50 | % | ALA2317819 | % | Homo sapiens | |||
| 4. |  [³H]naloxone | naloxone | INH | 0 | ALA3282289 | Active | % | Homo sapiens | ||||
| 5. | [³H]naloxone | naloxone | Activity | 0 | ALA3282288 | Active | Homo sapiens | |||||
| 6. |  ALA3274598 | 41 | Activity | 0 | ALA3282288 | Active | Homo sapiens | |||||
| 7. | ALA3274598 | 41 | Ratio IC50 | > | 10 | ALA3282290 | Homo sapiens | |||||
| 8. | ALA3274598 | 41 | IC50 | = | 5.7 | 10'-8M | ALA3282289 | 7.24 | nM | Homo sapiens | ||
| 9. | [³H]naloxone | naloxone | IC50 | = | 5.5 | nM | ALA3282287 | 8.26 | nM | Homo sapiens | ||
| 10. | ALA3274598 | 41 | IC50 | = | 5.3 | nM | ALA3282287 | 8.28 | nM | Homo sapiens | ||
| 11. |  ALA3274695 | Table II, R3C1 | FC | = | 2 | ALA3285644 | Homo sapiens | |||||
| 12. |  ALA3274694 | Table II, R2C1 | FC | = | 0.3 | ALA3285644 | Homo sapiens | |||||
| 13. |  ALA3274693 | Table II, R1C1 | FC | = | 50 | ALA3285644 | Homo sapiens | |||||
| 14. |  ALA3274696 | Table II, R4C1 | FC | = | 60 | ALA3285643 | Homo sapiens | |||||
| 15. | ALA3274694 | Table II, R2C1 | FC | = | 1000 | ALA3285643 | Homo sapiens | |||||
| 16. |  (S)-ARN2508 | (+)-10r | Activity | = | 15.5 | % | ALA3779679 | % | Homo sapiens | |||
| 17. |  GNE-8505 | 152 | Activity | > | 50 | % | ALA4120212 | % | Homo sapiens | |||
| 18. |  DLK-IN-1 | 165 | Activity | > | 50 | % | ALA4120212 | % | Homo sapiens | |||
| 19. |  ALA5179416 | (+)-16 | Activity | 0 | ALA5133298 | NA | Homo sapiens | |||||
| 20. |  ALA1270382 | SYK-3 | Activity | 0 | ALA5133298 | NA | Homo sapiens |
The page will load shortly, Thanks for your patience!