# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2420899 | 41 | INH | = | 29 | % | ALA2422073 | % | Homo sapiens | |||
2. | ALA2420900 | 42 | INH | = | 20 | % | ALA2422073 | % | Homo sapiens | |||
3. | ALA2420901 | 45 | INH | = | 28 | % | ALA2422073 | % | Homo sapiens | |||
4. | E1R | E1R, 4R,5S-2a | INH | = | -6 | % | ALA2393945 | % | Homo sapiens | |||
5. | ALA2071457 | (S)-24o | IC50 | > | 10 | uM | ALA2072602 | nM | Homo sapiens | |||
6. | ALA111612 | 10a | % inhibition | < | 10 | % | ALA4880267 | Not Active | % | Homo sapiens | ||
7. | ABT-100 | EUB0000289 | % inhibition | < | 10 | % | ALA4880188 | Not Active | % | Homo sapiens | ||
8. | ALA3697701 | BDBM161012 | % inhibition | -6 | % | ALA4880131 | Not Active | % | Homo sapiens | |||
9. | ALA213805 | CA224 | INH | 0 | ALA3375318 | Not Active | % | Homo sapiens | ||||
10. | ALA3335387 | 25 | IC50 | < | 10 | nM | ALA3384724 | nM | Homo sapiens | |||
11. | ALA3297762 | 15a | IC50 | > | 10 | uM | ALA3300947 | nM | Homo sapiens | |||
12. | ALA3298400 | 1 | IC50 | > | 10 | uM | ALA3300947 | nM | Homo sapiens | |||
13. | ALA3754043 | 7a | INH | 0 | ALA3757361 | Not Active | % | Homo sapiens | ||||
14. | Imatinib (STI571) | 1 | IC50 | = | 0.4 | uM | ALA3631066 | 6.40 | nM | Homo sapiens | ||
15. | ALA3086065 | 4b | IC50 | > | 50 | uM | ALA3090911 | nM | Homo sapiens | |||
16. | Sunitinib | 12b | IC50 | = | 0.08 | umol | ALA2066137 | 7.10 | nM | Homo sapiens | ||
17. | ALA1952211 | Ro-4383596, (-)-(S,S)-Enantiomer | IC50 | = | 33 | nM | ALA1952839 | 7.48 | nM | Homo sapiens | ||
18. | ALA1952210 | 6, Ro-4383596 | IC50 | = | 28 | nM | ALA1952839 | 7.55 | nM | Homo sapiens | ||
19. | ALA1952210 | 6, Ro-4383596 | IC50 | = | 33 | nM | ALA1952839 | 7.48 | nM | Homo sapiens | ||
20. | VEGFR2 Kinase Inhibitor I | 48 | IC50 | > | 100000 | nM | ALA937667 | nM | Homo sapiens |