# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798256 | 6a | Activity | = | 100 | % | ALA3802268 | % | Homo sapiens | |||
2. | ALA3758502 | 1 | INH | = | 14.1 | % | ALA3760632 | % | Homo sapiens | |||
3. | ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3747991 | nM | Homo sapiens | |||
4. | ALA3746293 | 23 | INH | = | -1.1 | % | ALA3751115 | % | Homo sapiens | |||
5. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | IC50 | = | 37 | uM | ALA3751415 | 4.43 | nM | Homo sapiens | ||
6. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | Kd | = | 2 | uM | ALA3751416 | 5.70 | nM | Homo sapiens | ||
7. | ALA3745744 | 2 | IC50 | = | 4.2 | uM | ALA3751415 | 5.38 | nM | Homo sapiens | ||
8. | ALA3747443 | 3 | IC50 | = | 30 | nM | ALA3751415 | 7.52 | nM | Homo sapiens | ||
9. | ALA3747095 | 4 | IC50 | = | 4 | nM | ALA3751415 | 8.40 | nM | Homo sapiens | ||
10. | ALA3746484 | 5 | IC50 | = | 150 | nM | ALA3751415 | 6.82 | nM | Homo sapiens | ||
11. | ALA3746157 | 6 | IC50 | = | 4 | nM | ALA3751415 | 8.40 | nM | Homo sapiens | ||
12. | ALA3628628 | 5 | INH | = | 0.04 | % | ALA3631290 | % | Homo sapiens | |||
13. | ALA3628627 | 4 | INH | = | 21.22 | % | ALA3631290 | % | Homo sapiens | |||
14. | ALA166031 | 3 | INH | = | 3.51 | % | ALA3631290 | % | Homo sapiens | |||
15. | ALA4530401 | EUB0000704 | % of control | = | 29.5 | % | ALA5213471 | % | Homo sapiens | |||
16. | ALA5178905 | (R)-STU104 | INH | < | 10 | % | ALA5165707 | % | Homo sapiens | |||
17. | ALA5178905 | (R)-STU104 | Kd | = | 3.61 | 10^-3/s | ALA5165705 | 10^-3/s | Homo sapiens | |||
18. | ALA5178905 | (R)-STU104 | Ka | = | 5.08 | 10^4/Ms | ALA5165704 | 10^4/Ms | Homo sapiens | |||
19. | ALA5178905 | (R)-STU104 | Kd | = | 71 | nM | ALA5165670 | 7.15 | nM | Homo sapiens | ||
20. | Imatinib (STI571) | 1 | Activity | 0 | ALA5120264 | Active | Homo sapiens |