# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Eplivanserin (mixture) | eplivanserin | Kd | = | 1.2 | nM | ALA5109946 | 8.92 | nM | Homo sapiens | ||
2. | ALA5204619 | [11C]MBL; [11C]70 | Ki | = | 0.5 | nM | ALA5109939 | 9.30 | nM | Homo sapiens | ||
3. | ALA221640 | [18F]79 | Ki | = | 760 | nM | ALA913684 | 6.12 | nM | Homo sapiens | ||
4. | ALA221652 | [18F]78 | Ki | = | 450 | nM | ALA913684 | 6.35 | nM | Homo sapiens | ||
5. | ALA2113241 | 23 | IC50 | > | 10000 | nmol/L | ALA870910 | nM | Homo sapiens | |||
6. | ALA210567 | (S)-6a | Ki | = | 2300 | nM | ALA860511 | 5.64 | nM | Homo sapiens | ||
7. | ALA210567 | (S)-6a | Ki | = | 1600 | nM | ALA860511 | 5.80 | nM | Homo sapiens | ||
8. | ALA210461 | 6b | Ki | = | 3500 | nM | ALA860511 | 5.46 | nM | Homo sapiens | ||
9. | ALA209876 | 6c | Ki | = | 470 | nM | ALA860511 | 6.33 | nM | Homo sapiens | ||
10. | ALA426863 | 6d | Ki | = | 1200 | nM | ALA860511 | 5.92 | nM | Homo sapiens | ||
11. | 2-Naphthalenecarboxamide, N-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)- | 39 | Ki | = | 840 | nM | ALA860511 | 6.08 | nM | Homo sapiens | ||
12. | ALA208847 | 4 | Ki | = | 2700 | nM | ALA860511 | 5.57 | nM | Homo sapiens | ||
13. | ALA202434 | 12h | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
14. | ALA1729 | cisapride | IC50 | = | 6.1 | nM | ALA858800 | 8.21 | nM | Homo sapiens | ||
15. | ALA2448165 | (R)-1C (SC-52491) | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
16. | ALA201946 | 13d | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
17. | ALA201878 | 13g | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
18. | ALA383577 | 13h | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
19. | SC 53116 | 1B | IC50 | > | 10000 | nM | ALA858800 | nM | Homo sapiens | |||
20. | ALA7257 | 11 | Activity | = | 26.1 | % | ALA861806 | % | Homo sapiens |