# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3127463 | (-)-36, enantiomer 1 | Ki | = | 740 | nM | ALA3129586 | 6.13 | nM | Homo sapiens | ||
2. | ALA3134464 | 21, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
3. | ALA3134465 | 25, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
4. | ALA3134466 | 22, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
5. | ALA2391037 | 8a-(2-chloro thiophene) | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
6. | ALA3134467 | 23, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
7. | ALA3134468 | 27, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
8. | ALA3134463 | 24, 1:1diastereomeric mixture | Ki | > | 100 | uM | ALA3135975 | nM | Homo sapiens | |||
9. | ALA143418 | 8 | IC50 | = | 800 | nM | ALA3134705 | 6.10 | nM | Homo sapiens | ||
10. | N-[(6-amino-2-methyl-3-pyridinyl)methyl]-2-[6-methyl-2-oxo-3-(2-phenylethylamino)-1-pyrazinyl]acetamide | L-375378 | IC50 | = | 1800 | nM | ALA3134705 | 5.75 | nM | Homo sapiens | ||
11. | ALA141889 | 20 | IC50 | = | 252 | nM | ALA3134705 | 6.60 | nM | Homo sapiens | ||
12. | ALA143024 | 25 | IC50 | = | 213 | nM | ALA3134705 | 6.67 | nM | Homo sapiens | ||
13. | ALA4568735 | EUB0000239 | % Inhibition | 0.8 | % | ALA4888326 | Not Active | % | Homo sapiens | |||
14. | ALA3640116 | BDBM100336 | % Ctrl | 108 | % | ALA4887752 | Not Active | % | Homo sapiens | |||
15. | ALA4588900 | EUB0001182 | % Inhibition of Control Values | 29.8 | % | ALA4882581 | % | Homo sapiens | ||||
16. | ALA5177478 | 105 | IC50 | = | 2.3 | uM | ALA5158488 | 5.64 | nM | Homo sapiens | ||
17. | ALA4594271 | BEROTRALSTAT | IC50 | = | 11 | uM | ALA4844459 | 4.96 | nM | Homo sapiens | ||
18. | ALA3289045 | 37 | Ki | > | 3000 | nM | ALA3294779 | nM | Homo sapiens | |||
19. | ALA3289044 | 36 | Ki | > | 3000 | nM | ALA3294779 | nM | Homo sapiens | |||
20. | ALA3289041 | 33 | Ki | > | 3000 | nM | ALA3294779 | nM | Homo sapiens |