# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288241 | B2 | IC50 | = | 950 | nM | ALA5238231 | 6.02 | nM | Homo sapiens | ||
2. | ALA5287062 | 40a | Ki | = | 0.279 | uM | ALA5230762 | 6.55 | nM | Homo sapiens | ||
3. | G1T38 | BDBM253941 | IC50 | = | 0.002 | uM | ALA5230719 | 8.70 | nM | Homo sapiens | ||
4. | AT7519 | 33 | IC50 | = | 10 | nM | ALA5230719 | 8.00 | nM | Homo sapiens | ||
5. | Palbociclib | 43(table 3) | IC50 | = | 16 | nM | ALA5230719 | 7.80 | nM | Homo sapiens | ||
6. | Flavopiridol | 1 | IC50 | = | 20 | nM | ALA5230719 | 7.70 | nM | Homo sapiens | ||
7. | Ribociclib | RIBOCICLIB | IC50 | = | 39 | nM | ALA5227268 | 7.41 | nM | Homo sapiens | ||
8. | Abemaciclib | ABEMACICLIB | IC50 | = | 10 | nM | ALA5227268 | 8.00 | nM | Homo sapiens | ||
9. | PF-06873600 | PF-06873600 | Ki | = | 0.16 | nM | ALA5227178 | 9.80 | nM | Homo sapiens | ||
10. | ALA4777981 | 63; A-1592668 | IC50 | = | 101 | nM | ALA5224484 | 7.00 | nM | Homo sapiens | ||
11. | ALA3668457 | BDBM167699 | IC50 | = | 298 | nM | ALA5224484 | 6.53 | nM | Homo sapiens | ||
12. | ALA5285499 | KI-ARv-03 | IC50 | > | 1200 | nM | ALA5224459 | nM | Homo sapiens | |||
13. | ALA5199065 | 55; KB-0742 | IC50 | > | 1200 | nM | ALA5224459 | nM | Homo sapiens | |||
14. | LDC 000067 | 5, LDC000067 | IC50 | > | 10000 | nM | ALA5224437 | nM | Homo sapiens | |||
15. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 6200 | nM | ALA5224410 | 5.21 | nM | Homo sapiens | ||
16. | voruciclib | VORUCICLIB | IC50 | = | 210 | nM | ALA5224410 | 6.68 | nM | Homo sapiens | ||
17. | Flavopiridol | 1 | IC50 | = | 60 | nM | ALA5224410 | 7.22 | nM | Homo sapiens | ||
18. | Abemaciclib | ABEMACICLIB | IC50 | = | 10 | nM | ALA5215110 | 8.00 | nM | Homo sapiens | ||
19. | Ribociclib | RIBOCICLIB | IC50 | = | 39 | nM | ALA5210389 | 7.41 | nM | Homo sapiens | ||
20. | Ribociclib | RIBOCICLIB | GI50 | = | 276 | nM | ALA5209971 | nM | Homo sapiens |