# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (±)-Methoxyverapamil hydrochloride | 4 | IC50 | = | 1.1 | 10'-8M | ALA2394916 | 7.96 | nM | Homo sapiens | ||
2. | (±)-Methoxyverapamil hydrochloride | 4 | Ki | = | 5.4 | 10'-9M | ALA2394916 | 8.27 | nM | Homo sapiens | ||
3. | ALA2069502 | 5a | IC50 | = | 1.9 | uM | ALA2072502 | 5.72 | nM | Homo sapiens | ||
4. | ALA2069501 | 4 | IC50 | = | 1526 | nM | ALA2072502 | 5.82 | nM | Homo sapiens | ||
5. | ALA2069500 | 3 | IC50 | = | 308 | nM | ALA2072502 | 6.51 | nM | Homo sapiens | ||
6. | BN-81,644 | 4k | IC50 | = | 128 | nM | ALA2072502 | 6.89 | nM | Homo sapiens | ||
7. | ALA2331983 | 52, isomer 2 | IC50 | = | 5.2 | uM | ALA2340381 | 5.28 | nM | Homo sapiens | ||
8. | ALA111612 | 10a | % inhibition | 29 | % | ALA4880304 | Not Active | % | Homo sapiens | |||
9. | ABT-100 | EUB0000289 | % inhibition | 10 | % | ALA4880228 | Not Active | % | Homo sapiens | |||
10. | ABT-100 | EUB0000289 | % inhibition | 37 | % | ALA4880228 | Not Active | % | Homo sapiens | |||
11. | ABT-100 | EUB0000289 | % inhibition | 60 | % | ALA4880228 | Slightly Active | % | Homo sapiens | |||
12. | ALA3697701 | BDBM161012 | % inhibition | 3 | % | ALA4880151 | Not Active | % | Homo sapiens | |||
13. | ALA4878564 | 28e | INH | = | 42 | % | ALA4845080 | % | Homo sapiens | |||
14. | ALA3912712 | 21s; BMS-963272 | INH | = | 24 | % | ALA4845080 | % | Homo sapiens | |||
15. | Omarigliptin (MK-3102) | OMARIGLIPTIN | Activity | 0 | ALA3239689 | Not Active | Homo sapiens | |||||
16. | PF 04418948 | 15, PF-04418948 | % inhibition | -5 | % | ALA4886961 | Not Active | % | Homo sapiens | |||
17. | PF 04418948 | 15, PF-04418948 | % inhibition | 6 | % | ALA4886960 | Not Active | % | Homo sapiens | |||
18. | PF 04418948 | 15, PF-04418948 | % inhibition | -3 | % | ALA4886959 | Not Active | % | Homo sapiens | |||
19. | ALA4536197 | EUB0000326 | % inhibition | -3 | % | ALA4886777 | Not Active | % | Homo sapiens | |||
20. | ALA4536197 | EUB0000326 | % inhibition | -5 | % | ALA4886761 | Not Active | % | Homo sapiens |