# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4444880 | 4 | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
2. | ALA4443665 | 3 | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
3. | ALA4441624 | 1a | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
4. | ALA4575627 | 1 | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
5. | ALA4470642 | 2a | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
6. | ALA4546687 | 2 | IC50 | > | 1000 | nM | ALA4413885 | nM | Homo sapiens | |||
7. | ALA4589933 | 16c; Diastereomeric mixture 4:1 | pIC50 | = | 7.1 | ALA4375394 | 7.10 | nM | Homo sapiens | |||
8. | ALA4239085 | 28u | pIC50 | = | 7.6 | ALA4375394 | 7.60 | nM | Homo sapiens | |||
9. | ALA4593110 | 16b; Diastereomeric mixture 3:1 | pIC50 | = | 6.2 | ALA4375394 | 6.20 | nM | Homo sapiens | |||
10. | ALA4446267 | 15b | pIC50 | = | 6.8 | ALA4375394 | 6.80 | nM | Homo sapiens | |||
11. | ALA4446786 | 16a; Diastereomeric mixture 5:1 | pIC50 | = | 6.6 | ALA4375394 | 6.60 | nM | Homo sapiens | |||
12. | ALA4238909 | 28c | pIC50 | = | 7.3 | ALA4375394 | 7.30 | nM | Homo sapiens | |||
13. | ALA4516070 | 14 | pIC50 | < | 5 | ALA4375394 | nM | Homo sapiens | ||||
14. | ALA4573716 | 8 | pIC50 | = | 6 | ALA4375394 | 6.00 | nM | Homo sapiens | |||
15. | (3S)-3-(3-(3,5-Dimethyl-1H-pyrazol-1-yl)phenyl)-4-((1S,3R)-1-methyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-ium-1-yl)butanoate | 7 | pIC50 | = | 6.3 | ALA4375394 | 6.30 | nM | Homo sapiens | |||
16. | ALA4246089 | 28h.HCl | pIC50 | = | 6.9 | ALA4375394 | 6.90 | nM | Homo sapiens | |||
17. | ALA4448207 | 5 | pIC50 | = | 7.1 | ALA4375389 | 7.10 | nM | Homo sapiens | |||
18. | CWHM12 | 34, CWHM12 | IC50 | = | 61 | nM | ALA4375379 | 7.21 | nM | Homo sapiens | ||
19. | ALA4246089 | 28h.HCl | pKi | = | 8 | ALA4375379 | 8.00 | nM | Homo sapiens | |||
20. | GLPG 0187 | 33, GLPG0187 | IC50 | = | 2 | nM | ALA4375384 | 8.70 | nM | Homo sapiens |