# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA370148 | 273 (Truncated brevetoxin B) | Binding | = | 18 | nM | ALA872318 | nM | Homo sapiens | |||
2. | ALA370148 | 273 (Truncated brevetoxin B) | IC50 | > | 10000 | nM | ALA880612 | nM | Homo sapiens | |||
3. | Brevetoxin2 (PbTx-2) | 272 (Brevetoxin B) | Binding | = | 18 | nM | ALA872318 | nM | Homo sapiens | |||
4. | Brevetoxin2 (PbTx-2) | 272 (Brevetoxin B) | IC50 | = | 15.02 | nM | ALA880612 | 7.82 | nM | Homo sapiens | ||
5. | ALA370148 | 273 (Truncated brevetoxin B) | Binding | = | 18 | nM | ALA872318 | nM | Homo sapiens | |||
6. | ALA370148 | 273 (Truncated brevetoxin B) | IC50 | > | 10000 | nM | ALA880607 | nM | Homo sapiens | |||
7. | Brevetoxin2 (PbTx-2) | 272 (Brevetoxin B) | Binding | = | 18 | nM | ALA872318 | nM | Homo sapiens | |||
8. | Brevetoxin2 (PbTx-2) | 272 (Brevetoxin B) | IC50 | = | 15.02 | nM | ALA880607 | 7.82 | nM | Homo sapiens | ||
9. | ALA55922 | 3a | IC50 | = | 1000 | uM | ALA749469 | nM | Homo sapiens | |||
10. | ALA52359 | 3c | IC50 | = | 0.5 | uM | ALA749469 | 6.30 | nM | Homo sapiens | ||
11. | ALA298513 | 4a | IC50 | = | 80 | uM | ALA749469 | 4.10 | nM | Homo sapiens | ||
12. | ALA52258 | 3b | IC50 | = | 200 | uM | ALA749469 | nM | Homo sapiens | |||
13. | ALA296366 | 3d | IC50 | = | 5 | uM | ALA749469 | 5.30 | nM | Homo sapiens | ||
14. | ALA55733 | 4b | IC50 | = | 4 | uM | ALA749469 | 5.40 | nM | Homo sapiens | ||
15. | Tetracaine | 3 | IC50 | = | 0.4 | uM | ALA749469 | 6.40 | nM | Homo sapiens | ||
16. | ALA145968 | 10 | IC50 | > | 25 | uM | ALA752430 | nM | Homo sapiens | |||
17. | ALA539841 | 13 | IC50 | > | 25 | uM | ALA752430 | nM | Homo sapiens | |||
18. | ALA422495 | 14 | IC50 | > | 25 | uM | ALA752430 | nM | Homo sapiens | |||
19. | ALA145968 | 10 | IC50 | > | 25 | uM | ALA752430 | nM | Homo sapiens | |||
20. | Cns-5161 | 1 | IC50 | = | 1.75 | uM | ALA752430 | 5.76 | nM | Homo sapiens |