# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NMS-E973 | 18, NMS-E973 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
2. | ALA2443138 | 30 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
3. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
4. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
5. | ALA1940990 | 23 | INH | < | 35 | % | ALA1943334 | % | Homo sapiens | |||
6. | ALA1940987 | 20 | INH | < | 35 | % | ALA1943334 | % | Homo sapiens | |||
7. | ALA1940981 | 14 | INH | < | 35 | % | ALA1943334 | % | Homo sapiens | |||
8. | ALA1940980 | 13 | INH | < | 35 | % | ALA1943334 | % | Homo sapiens | |||
9. | ALA1834330 | 43 | INH | < | 35 | % | ALA1837573 | % | Homo sapiens | |||
10. | ALA1834324 | 37 | INH | < | 35 | % | ALA1837573 | % | Homo sapiens | |||
11. | ALA1834323 | 36 | INH | < | 35 | % | ALA1837573 | % | Homo sapiens | |||
12. | ALA1834318 | 28 | INH | < | 35 | % | ALA1837573 | % | Homo sapiens | |||
13. | ALA1834114 | 11 | INH | = | 48.3 | % | ALA1837573 | % | Homo sapiens | |||
14. | ALA373101 | 12 | IC50 | = | 1.3 | nM | ALA883697 | 8.89 | nM | Homo sapiens | ||
15. | ALA364955 | 3 | IC50 | = | 2.3 | nM | ALA883697 | 8.64 | nM | Homo sapiens | ||
16. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | IC50 | = | 1 | nM | ALA883697 | 9.00 | nM | Homo sapiens | ||
17. | Ponatinib (AP24534) | 20g, AP24534 | INH | 0 | ALA1176910 | Active | % | Homo sapiens | ||||
18. | Ponatinib (AP24534) | 20g, AP24534 | INH | 0 | ALA1176909 | Active | % | Homo sapiens | ||||
19. | ALA311129 | 28 | IC50 | > | 100 | uM | ALA846549 | nM | Homo sapiens | |||
20. | ALA308582 | 12 | IC50 | = | 99 | uM | ALA846549 | 4.00 | nM | Homo sapiens |