# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N-[(1R)-1-(N'-cyano-N,N'-dimethylhydrazinecarbonyl)-2-(2-methylpropanesulfonyl)ethyl]benzamide | (R)-26 | Ki | = | 21 | nM | ALA2156365 | 7.68 | nM | Homo sapiens | ||
2. | ALA2153172 | (R)-22 | Ki | > | 40 | uM | ALA2157194 | nM | Homo sapiens | |||
3. | ALA2153171 | (+/-)-16 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
4. | ALA2153170 | (+/-)-15 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
5. | ALA2153169 | (+/-)-14 | Ki | = | 3.2 | uM | ALA2157194 | 5.50 | nM | Homo sapiens | ||
6. | ALA2153168 | (+/-)-13 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
7. | ALA2153167 | (+/-)-12 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
8. | ALA2153166 | (+/-)-11 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
9. | ALA2153165 | (+/-)-10 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
10. | ALA2153164 | (+/-)-9 | Ki | > | 4 | uM | ALA2157194 | nM | Homo sapiens | |||
11. | ALA2153163 | (+/-)-8 | Ki | > | 40 | uM | ALA2157194 | nM | Homo sapiens | |||
12. | ALA2153162 | (+/-)-7 | Ki | > | 40 | uM | ALA2157194 | nM | Homo sapiens | |||
13. | ALA3586467 | 231 | IP | = | 3142 | nM | ALA3586962 | nM | Homo sapiens | |||
14. | ALA3586466 | 110 | IP | = | 3333 | nM | ALA3586962 | nM | Homo sapiens | |||
15. | ALA3586465 | 19 | IP | = | 851 | nM | ALA3586962 | nM | Homo sapiens | |||
16. | ALA3586464 | 1 | IP | = | 1000 | nM | ALA3586962 | nM | Homo sapiens | |||
17. | ALA4127793 | E-64 | INH | = | 50 | % | ALA4686589 | % | Homo sapiens | |||
18. | ALA3289242 | 38 | INH | 0 | ALA4686583 | Not Active | % | Homo sapiens | ||||
19. | ALA4751760 | 31 | INH | 0 | ALA4686583 | Not Active | % | Homo sapiens | ||||
20. | ALA4799416 | 30 | INH | 0 | ALA4686583 | Not Active | % | Homo sapiens |