# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-Methylmellein | 7 | IC50 | = | 1.06 | uM | ALA4393411 | 5.97 | nM | Mus musculus | ||
2. | ALA4545549 | 69.HCl | Activity | = | 31.3 | % | ALA4325546 | % | Mus musculus | |||
3. | ALA4447820 | 100.HCl | Activity | = | 59.4 | % | ALA4325546 | % | Mus musculus | |||
4. | ALA554000 | 1 | Inhibition | = | 8.5 | % | ALA821702 | % | Mus musculus | |||
5. | ALA97993 | 10 | Inhibition | = | 16 | % | ALA821701 | % | Mus musculus | |||
6. | Selegiline | (-)-Deprenyl | Activity | = | 1.36 | nM | ALA731240 | nM | Mus musculus | |||
7. | Selegiline | (-)-Deprenyl | Activity | = | 0.84 | nM | ALA731240 | nM | Mus musculus | |||
8. | ALA343006 | 16 ; carbamate(S) | Activity | = | 3.75 | nM | ALA731239 | nM | Mus musculus | |||
9. | ALA145281 | 16 ; carbamate(R) | Activity | = | 1.36 | nM | ALA731239 | nM | Mus musculus | |||
10. | R-(-)-N-Demethyl deprenyl | (R)nordeprenyl | Activity | = | 1.31 | nM | ALA731240 | nM | Mus musculus | |||
11. | ALA2028089 | (R)(-)2 | Inhibition | = | 14 | % | ALA731246 | % | Mus musculus | |||
12. | ALA2028089 | (R)(-)2 | ED50 | = | 54 | uM kg-1 | ALA731243 | umol.kg-1 | Mus musculus | |||
13. | ALA2028089 | (R)(-)2 | ED50 | > | 72 | uM kg-1 | ALA731241 | umol.kg-1 | Mus musculus | |||
14. | Selegiline | (-)-Deprenyl | Inhibition | = | 25 | % | ALA731246 | % | Mus musculus | |||
15. | Selegiline | (-)-Deprenyl | ED50 | = | 2 | uM kg-1 | ALA731243 | umol.kg-1 | Mus musculus | |||
16. | Selegiline | (-)-Deprenyl | ED50 | > | 89 | uM kg-1 | ALA731241 | umol.kg-1 | Mus musculus | |||
17. | ALA9068 | 9 | Inhibition | = | 7 | % | ALA731246 | % | Mus musculus | |||
18. | ALA9068 | 9 | ED50 | = | 11 | uM kg-1 | ALA731243 | umol.kg-1 | Mus musculus | |||
19. | ALA9068 | 9 | ED50 | > | 38 | uM kg-1 | ALA731241 | umol.kg-1 | Mus musculus | |||
20. | ALA276375 | 2 | Inhibition | = | 18 | % | ALA731247 | % | Mus musculus |